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Found 7 Enz. Inhib. hit(s) with all data for entry = 50006421
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Michigan Medical School

Curated by ChEMBL
LigandPNGBDBM50048893((2R,3R,11bR)-3-Isobutyl-9,10-dimethoxy-2-methyl-1,...)
Affinity DataKi:  2.60nMAssay Description:Compound was tested in vitro for the inhibition of [3H]- Methoxytetrabenazine binding to rat brain vesicular monoamine transporter 2 (VMAT2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Michigan Medical School

Curated by ChEMBL
LigandPNGBDBM50048891((3R,11bR)-3-Isobutyl-9,10-dimethoxy-1,3,4,6,7,11b-...)
Affinity DataKi:  8.10nMAssay Description:Compound was tested in vitro for the inhibition of [3H]- Methoxytetrabenazine binding to rat brain vesicular monoamine transporter 2 (VMAT2)More data for this Ligand-Target Pair
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Michigan Medical School

Curated by ChEMBL
LigandPNGBDBM50048892((2S,3R,11bR)-3-Isobutyl-9,10-dimethoxy-2-methyl-1,...)
Affinity DataKi:  12nMAssay Description:Compound was tested in vitro for the inhibition of [3H]- Methoxytetrabenazine binding to rat brain vesicular monoamine transporter 2 (VMAT2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Michigan Medical School

Curated by ChEMBL
LigandPNGBDBM50048895((2S,3R,11bR)-2,3-Diisobutyl-9,10-dimethoxy-1,3,4,6...)
Affinity DataKi:  33nMAssay Description:Compound was tested in vitro for the inhibition of [3H]- Methoxytetrabenazine binding to rat brain vesicular monoamine transporter 2 (VMAT2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Michigan Medical School

Curated by ChEMBL
LigandPNGBDBM50048897((2S,3R,11bR)-2-Ethyl-3-isobutyl-9,10-dimethoxy-1,3...)
Affinity DataKi:  42nMAssay Description:Compound was tested in vitro for the inhibition of [3H]- Methoxytetrabenazine binding to rat brain vesicular monoamine transporter 2 (VMAT2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Michigan Medical School

Curated by ChEMBL
LigandPNGBDBM50048894((2S,3R,11bR)-3-Isobutyl-9,10-dimethoxy-2-propyl-1,...)
Affinity DataKi:  84nMAssay Description:Compound was tested in vitro for the inhibition of [3H]- Methoxytetrabenazine binding to rat brain vesicular monoamine transporter 2 (VMAT2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Michigan Medical School

Curated by ChEMBL
LigandPNGBDBM50048896((2S,3R,11bR)-2-tert-Butyl-3-isobutyl-9,10-dimethox...)
Affinity DataKi:  136nMAssay Description:Compound was tested in vitro for the inhibition of [3H]- Methoxytetrabenazine binding to rat brain vesicular monoamine transporter 2 (VMAT2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed