Compile Data Set for Download or QSAR
maximum 50k data
Found 41 Enz. Inhib. hit(s) with all data for entry = 50007429
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063215(CHEMBL158859 | [3-(2-Chloro-benzyl)-3H-[1,2,3]tria...)
Affinity DataKi:  21nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50408698(CHEMBL2112325)
Affinity DataKi:  39nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063204(CHEMBL161711 | [3-(2-Chloro-benzyl)-3H-[1,2,3]tria...)
Affinity DataKi:  43nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063190(CHEMBL159178 | [3-(2-Chloro-benzyl)-3H-[1,2,3]tria...)
Affinity DataKi:  73nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063184(CHEMBL161051 | [3-(2-Chloro-benzyl)-3H-[1,2,3]tria...)
Affinity DataKi:  102nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063189(CHEMBL158598 | [3-(2-Chloro-benzyl)-3H-[1,2,3]tria...)
Affinity DataKi:  119nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063198((3-Benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)...)
Affinity DataKi:  121nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063185((3-Benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)...)
Affinity DataKi:  127nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063180(CHEMBL347834 | Cyclopentyl-(3-phenethyl-3H-[1,2,3]...)
Affinity DataKi:  176nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063210(CHEMBL161326 | Cyclohexyl-(3-phenethyl-3H-[1,2,3]t...)
Affinity DataKi:  216nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063217((4-Nitro-benzyl)-(3-phenethyl-3H-[1,2,3]triazolo[4...)
Affinity DataKi:  245nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50408699(CHEMBL2110165)
Affinity DataKi:  274nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063211((3-Benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)...)
Affinity DataKi:  438nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063206((3-Benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)...)
Affinity DataKi:  443nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063194((3-Benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)...)
Affinity DataKi:  463nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063195(CHEMBL161425 | [3-(2-Chloro-benzyl)-3H-[1,2,3]tria...)
Affinity DataKi:  468nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063191((3-Benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)...)
Affinity DataKi:  502nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063199((3-Benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)...)
Affinity DataKi:  575nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063200((3-Benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)...)
Affinity DataKi:  770nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063208(CHEMBL349650 | N-[3-(2-Chloro-benzyl)-3H-[1,2,3]tr...)
Affinity DataKi: >1.00E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063213(CHEMBL350078 | [3-(2-Chloro-benzyl)-3H-[1,2,3]tria...)
Affinity DataKi: >1.00E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063186((4-Amino-benzyl)-[3-(2-chloro-benzyl)-3H-[1,2,3]tr...)
Affinity DataKi: >1.00E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063214((3-Benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)...)
Affinity DataKi: >1.00E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063187((3-Benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)...)
Affinity DataKi: >1.00E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063182(CHEMBL161766 | [3-(2-Chloro-benzyl)-3H-[1,2,3]tria...)
Affinity DataKi: >1.00E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063203((3-Benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)...)
Affinity DataKi:  1.10E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063209(CHEMBL158483 | [2-(4-Amino-phenyl)-ethyl]-(3-benzy...)
Affinity DataKi:  1.54E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063201((3-Phenethyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-...)
Affinity DataKi:  1.67E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063188(CHEMBL162531 | [3-(2-Chloro-benzyl)-3H-[1,2,3]tria...)
Affinity DataKi:  1.83E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063205((3-Phenethyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-...)
Affinity DataKi:  2.20E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063192((3-Nitro-phenyl)-(3-phenethyl-3H-[1,2,3]triazolo[4...)
Affinity DataKi:  2.25E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063202((1-Methyl-2-phenyl-ethyl)-(3-phenethyl-3H-[1,2,3]t...)
Affinity DataKi:  2.49E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063212((3-Benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)...)
Affinity DataKi:  2.79E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063179(CHEMBL351691 | [3-(2-Chloro-benzyl)-3H-[1,2,3]tria...)
Affinity DataKi:  3.30E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063183((3-Chloro-phenyl)-(3-phenethyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  3.32E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063181(CHEMBL162247 | [3-(2-Chloro-benzyl)-3H-[1,2,3]tria...)
Affinity DataKi:  4.26E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063193((3-Phenethyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-...)
Affinity DataKi:  4.38E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063197(CHEMBL158423 | [3-(2-Chloro-benzyl)-3H-[1,2,3]tria...)
Affinity DataKi:  5.88E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50063207(CHEMBL157641 | N-(3-Benzyl-3H-[1,2,3]triazolo[4,5-...)
Affinity DataKi:  6.70E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063196(CHEMBL161227 | N-(3-Phenethyl-3H-[1,2,3]triazolo[4...)
Affinity DataKi:  7.20E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063216((4-Amino-benzyl)-(3-benzyl-3H-[1,2,3]triazolo[4,5-...)
Affinity DataKi:  9.50E+3nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed