Reaction Details Report a problem with these data
Target
Alpha-2C adrenergic receptor
Ligand
BDBM81802
Substrate
n/a
Ki
804±n/a nM
Comments
PDSP_505
Citation
 Blaxall, HS; Murphy, TJ; Baker, JC; Ray, C; Bylund, DB Characterization of the alpha-2C adrenergic receptor subtype in the opossum kidney and in the OK cell line. J Pharmacol Exp Ther 259:323-9 (1991) [PubMed] 
Target
Name:
Alpha-2C adrenergic receptor
Synonyms:
ADRA2C | adrenergic Alpha2C
Type:
Enzyme Catalytic Domain
Mol. Mass.:
27257.01
Organism:
OK
Description:
adrenergic Alpha2C ADRA2C OK::G3GWB4
Residue:
230
Sequence:
MAYWYFGQVWCGVYLALDVLFCTSSIVHLCAISLDRYWSVTQAVEYNLKRTPRRVKATIVAVWLISAVISFPPLVSFYRRSDGAAYPQCGLNDETWYILSSCIGSFFAPCLIMGLVYARIYRFFLSRRRRARSSVCRRKVAQAREKRFTFVLAVVMGVFVLCWFPFFFSYSLYGICREACQLPEPLFKFFFWIGYCKSSLNPVIYTVFNQDFRRSFKHILFRRRRRGFRQ
  
Inhibitor
Name:
BDBM81802
Synonyms:
CAS_81382-52-7 | CGS-10746B | CGS10746B | PENTIAPINE MALEATE
Type:
Small organic molecule
Emp. Form.:
C15H17N5S
Mol. Mass.:
299.394
SMILES:
CN1CCN(CC1)C1=Nc2ccccc2Sc2nccn12 |t:8|
Structure:
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