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Target
Pituitary adenylate cyclase-activating polypeptide
Ligand
BDBM81827
Substrate
n/a
Ki
680±n/a nM
Comments
PDSP_2614
Citation
 Schäfer, H; Schwarzhoff, R; Creutzfeldt, W; Schmidt, WE Characterization of a guanosine-nucleotide-binding-protein-coupled receptor for pituitary adenylate-cyclase-activating polypeptide on plasma membranes from rat brain. Eur J Biochem 202:951-8 (1991) [PubMed]  Article 
Target
Name:
Pituitary adenylate cyclase-activating polypeptide
Synonyms:
Adcyap1 | PACAP | PACAP-27 | PACAP-38 | PACA_RAT | Pituitary adenylate cyclase-activating polypeptide
Type:
Enzyme Catalytic Domain
Mol. Mass.:
19565.66
Organism:
RAT
Description:
PACAP 0 RAT::P13589
Residue:
175
Sequence:
MTMCSGARLALLVYGIIMHNSVSCSPAAGLSFPGIRPEEEAYDQDGNPLQDFYDWDPPGAGSPASALRDAYALYYPADRRDVAHEILNEAYRKVLDQLSARKYLQSMVARGMGENLAAAAVDDRAPLTKRHSDGIFTDSYSRYRKQMAVKKYLAAVLGKRYKQRVKNKGRRIAYL
  
Inhibitor
Name:
BDBM81827
Synonyms:
GuoPP[NH]P
Type:
Small organic molecule
Emp. Form.:
C11H16N5O14P3
Mol. Mass.:
535.1911
SMILES:
Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H](COP(O)(=O)OP2(=O)OCOP(O)(=O)O2)[C@@H](O)[C@H]1O
Structure:
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