Reaction Details Report a problem with these data
Target
Virulence factor transcriptional regulator MvfR
Ligand
BDBM50512173
Substrate
n/a
Meas. Tech.
ChEMBL_1848045 (CHEMBL4348586)
IC50
3900±n/a nM
Citation
Soheili, V; Tajani, AS; Ghodsi, R; Bazzaz, BSF Anti-PqsR compounds as next-generation antibacterial agents against Pseudomonas aeruginosa: A review. Eur J Med Chem 172:26-35 (2019) [PubMed] Article
More Info.:
Target
Name:
Virulence factor transcriptional regulator MvfR
Synonyms:
Transcriptional regulator MvfR
Type:
PROTEIN
Mol. Mass.:
37217.11
Organism:
Pseudomonas aeruginosa PA14
Description:
ChEMBL_107649
Residue:
332
Sequence:
MPIHNLNHVNMFLQVIASGSISSAARILRKSHTAVSSAVSNLEIDLCVELVRRDGYKVEPTEQALRLIPYMRSLLNYQQLIGDIAFNLNKGPRNLRVLLDTAIPPSFCDTVSSVLLDDFNMVSLIRTSPADSLATIKQDNAEIDIAITIDEELKISRFNQCVLGYTKAFVVAHPQHPLCNASLHSIASLANYRQISLGSRSGQHSNLLRPVSDKVLFVENFDDMLRLVEAGVGWGIAPHYFVEERLRNGTLAVLSELYEPGGIDTKVYCYYNTALESERSFLRFLESARQRLRELGRQRFDDAPAWQPSIVETAQRRSGPKALAYRQRAAPE