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Target
G-protein coupled receptor 84
Ligand
BDBM50239172
Substrate
n/a
Meas. Tech.
ChEMBL_2057173 (CHEMBL4712174)
EC50
295±n/a nM
Citation
 Chen, LH; Zhang, Q; Xie, X; Nan, FJ Modulation of the G-Protein-Coupled Receptor 84 (GPR84) by Agonists and Antagonists. J Med Chem 63:15399-15409 (2020) [PubMed]  Article 
Target
Name:
G-protein coupled receptor 84
Synonyms:
G-protein coupled receptor 84 | GPR84_MOUSE | Gpr84
Type:
PROTEIN
Mol. Mass.:
43740.69
Organism:
Mus musculus
Description:
ChEMBL_119136
Residue:
396
Sequence:
MWNSSDANFSCYHESVLGYRYFAVIWGVAVAVTGTVGNVLTLLALAIRPKLRTRFNLLIANLTLADLLYCTLLQPFSVDTYLHLHWRTGAVFCRIFGLLLFTSNSVSILTLCLIALGRYLLIAHPKLFPQVFSAKGIVLALVGSWVVGVTSFAPLWNVFVLVPVVCTCSFDRMRGRPYTTILMGIYFVLGLSSVGVFYCLIHRQVKRAARALDQYGLHQASIRSHQVAGTQEAMPGHFQELDSGVASRGPSEGISSEPVSAATTQTLEGDSSEAGGQGIRKAAQQIAERSLPEVHRKPRETAGARRATDAPSEFGKVTRMCFAVFLCFALSYIPFLLLNILDARGRAPRVVHMVAANLTWLNSCINPVLYAAMNRQFRHAYGSILKRGPQSFRRFH
  
Inhibitor
Name:
BDBM50239172
Synonyms:
CHEMBL4088884
Type:
Small organic molecule
Emp. Form.:
C17H10F4N2
Mol. Mass.:
318.2683
SMILES:
Fc1cc(F)c2[nH]cc(Cc3c[nH]c4c(F)cc(F)cc34)c2c1
Structure:
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