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Target
Mu-type opioid receptor
Ligand
BDBM50310292
Substrate
n/a
Meas. Tech.
ChEMBL_607972 (CHEMBL1071742)
Ki
24±n/a nM
Citation
 Imaide, S; Fujii, H; Watanabe, A; Nemoto, T; Nakajima, M; Nakao, K; Mochizuki, H; Nagase, H Investigation of Beckett-Casy model 1: synthesis of novel 16,17-seco-naltrexone derivatives and their pharmacology. Bioorg Med Chem Lett 20:1055-8 (2010) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50310292
Synonyms:
CHEMBL604522 | KNT-5
Type:
Small organic molecule
Emp. Form.:
C21H25NO4
Mol. Mass.:
355.4275
SMILES:
CN(CC1CC1)[C@@H]1Cc2ccc(O)c3O[C@H]4C(=O)CC[C@@]11OCC[C@]41c23 |r|
Structure:
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