Reaction Details Report a problem with these data
Target
Succinate dehydrogenase cytochrome b560 subunit, mitochondrial
Ligand
BDBM50079600
Substrate
n/a
Meas. Tech.
ChEMBL_1472196 (CHEMBL3418827)
Ki
327±n/a nM
Citation
 Xiong, L; Zhu, XL; Shen, YQ; Wishwajith, WK; Li, K; Yang, GF Discovery of N-benzoxazol-5-yl-pyrazole-4-carboxamides as nanomolar SQR inhibitors. Eur J Med Chem 95:424-34 (2015) [PubMed]  Article 
Target
Name:
Succinate dehydrogenase cytochrome b560 subunit, mitochondrial
Synonyms:
C560_PIG | CYBL | SDHC | Succinate dehydrogenase cytochrome b560 subunit, mitochondrial | Succinate-ubiquinone oxidoreductase cytochrome B large subunit
Type:
PROTEIN
Mol. Mass.:
18529.95
Organism:
Sus scrofa
Description:
ChEMBL_106708
Residue:
169
Sequence:
MAALLLRHVGRHCLRAHLSPQLCIRNAVPLGTTAKEEMERFWNKNLGSNRPLSPHITIYRWSLPMAMSICHRGTGIALSAGVSLFGLSALLLPGNFESHLELVKSLCLGPTLIYTAKFGIVFPLMYHTWNGIRHLIWDLGKGLTIPQLTQSGVVVLILTVLSSVGLAAM
  
Inhibitor
Name:
BDBM50079600
Synonyms:
CHEBI:83138 | PENTHIOPYRAD
Type:
Small organic molecule
Emp. Form.:
C16H20F3N3OS
Mol. Mass.:
359.41
SMILES:
CC(C)CC(C)c1sccc1NC(=O)c1cn(C)nc1C(F)(F)F
Structure:
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