Reaction Details Report a problem with these data
Target
Histamine H2 receptor
Ligand
BDBM82472
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_456
Citation
 Baxter, GS Novel discriminatory ligands for 5-HT2B receptors. Behav Brain Res 73:149-52 (1996) [PubMed]  Article 
Target
Name:
Histamine H2 receptor
Synonyms:
HISTAMINE H2 | HRH2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40972.37
Organism:
RABBIT
Description:
HISTAMINE H2 HRH2 RABBIT::G1TWL8
Residue:
367
Sequence:
MEPNDTANDTASSSCLESTAFKVTLSVVLTILILITAAGNVVVCLAVGLNRRLRSLTNCFIVSLAITDLLLGLLVLPFSAIYQLSCRWSFGKVFCNIYISLDVMLCTASILNLFMISIDRYCAVTDPLRYPVLVTPGRVTISLVSIWVISITLSFLSIHLGWNSRNTTSEGHHTSPKCKFQVNEVYGLVDGLVTFYLPLLIMCVTYYRIFKIAREQARRINHISSWQAATIREHKATVTLAAVMGAFIVCWFPYFTTFVYRGLKGDDAINEVVEAVVLWLGYANSALNPILYAALNRDFRNAYQQLFCCRLAGRGSHETCLRFNNALLPKSQSQEPRRQEEKPLKLQVWSGTEATAPQGATDRVFGE
  
Inhibitor
Name:
BDBM82472
Synonyms:
BW-723C86 | CAS_5311036 | NSC_5311036
Type:
Small organic molecule
Emp. Form.:
C16H18N2OS
Mol. Mass.:
286.392
SMILES:
CC(N)Cc1c[nH]c2ccc(OCc3cccs3)cc12
Structure:
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