Reaction Details
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Somatostatin receptor type 5
Ligand
BDBM85230
Substrate
n/a
Ki
0.27±n/a nM
Comments
PDSP_3571
Citation
Meyerhof, W The elucidation of somatostatin receptor functions: a current view. Rev Physiol Biochem Pharmacol 133:55-108 (1998) [PubMed] Article More Info.:
Target
Name:
Somatostatin receptor type 5
Synonyms:
SOMATOSTATIN SST5 | SS-5-R | SS5-R | SS5R | SSR5_HUMAN | SSTR5 | Somatostatin receptor type 5 (SSTR5)
Type:
Enzyme
Mol. Mass.:
39218.02
Organism:
Homo sapiens (Human)
Description:
P35346
Residue:
364
Sequence:
MEPLFPASTPSWNASSPGAASGGGDNRTLVGPAPSAGARAVLVPVLYLLVCAAGLGGNTLVIYVVLRFAKMKTVTNIYILNLAVADVLYMLGLPFLATQNAASFWPFGPVLCRLVMTLDGVNQFTSVFCLTVMSVDRYLAVVHPLSSARWRRPRVAKLASAAAWVLSLCMSLPLLVFADVQEGGTCNASWPEPVGLWGAVFIIYTAVLGFFAPLLVICLCYLLIVVKVRAAGVRVGCVRRRSERKVTRMVLVVVLVFAGCWLPFFTVNIVNLAVALPQEPASAGLYFFVVILSYANSCANPVLYGFLSDNFRQSFQKVLCLRKGSGAKDADATEPRPDRIRQQQEATPPAHRAAANGLMQTSKL
Inhibitor
Name:
BDBM85230
Synonyms:
BIM 23313
Type:
Small organic molecule
Emp. Form.:
C54H69N11O9S2
Mol. Mass.:
1080.324
SMILES:
CC(O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1ccccc1)NC(=O)C(Cc1ccccc1)NC(=O)C(N)CS)C(=O)NC(Cc1ccccc1)C(=O)NC(CS)C(N)=O
Structure:
