Reaction Details Report a problem with these data
Target
Norepinephrine transporter
Ligand
BDBM30130
Substrate
n/a
Ki
119±n/a nM
Comments
PDSP_830
Citation
 Béïque, JC; Lavoie, N; de Montigny, C; Debonnel, G Affinities of venlafaxine and various reuptake inhibitors for the serotonin and norepinephrine transporters. Eur J Pharmacol 349:129-32 (1998) [PubMed]  Article 
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
  
Inhibitor
Name:
BDBM30130
Synonyms:
CHEMBL1201082 | CHEMBL41 | Fluoxetin | Fluoxetine | Prozac | US9120771, Fluoxetine | cid_62857
Type:
Small organic molecule
Emp. Form.:
C17H18F3NO
Mol. Mass.:
309.3261
SMILES:
CNCCC(Oc1ccc(cc1)C(F)(F)F)c1ccccc1
Structure:
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