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Target
C-terminal-binding protein 2
Ligand
BDBM154570
Substrate
n/a
Meas. Tech.
CtBP2 ITC
pH
8.5±0
Kd
1.30e+3± 7e+1 nM
Citation
Hilbert, BJ; Morris, BL; Ellis, KC; Paulsen, JL; Schiffer, CA; Grossman, SR; Royer, WE Structure-guided design of a high affinity inhibitor to human CtBP. ACS Chem Biol 10:1118-27 (2015) [PubMed] Article
More Info.:
Target
Name:
C-terminal-binding protein 2
Synonyms:
C-terminal-binding protein 2 | C-terminal-binding protein 2 (CtBP2) | CTBP2 | CTBP2_HUMAN
Type:
Protein
Mol. Mass.:
48948.33
Organism:
Homo sapiens (Human)
Description:
P56545
Residue:
445
Sequence:
MALVDKHKVKRQRLDRICEGIRPQIMNGPLHPRPLVALLDGRDCTVEMPILKDLATVAFCDAQSTQEIHEKVLNEAVGAMMYHTITLTREDLEKFKALRVIVRIGSGYDNVDIKAAGELGIAVCNIPSAAVEETADSTICHILNLYRRNTWLYQALREGTRVQSVEQIREVASGAARIRGETLGLIGFGRTGQAVAVRAKAFGFSVIFYDPYLQDGIERSLGVQRVYTLQDLLYQSDCVSLHCNLNEHNHHLINDFTIKQMRQGAFLVNAARGGLVDEKALAQALKEGRIRGAALDVHESEPFSFAQGPLKDAPNLICTPHTAWYSEQASLEMREAAATEIRRAITGRIPESLRNCVNKEFFVTSAPWSVIDQQAIHPELNGATYRYPPGIVGVAPGGLPAAMEGIIPGGIPVTHNLPTVAHPSQAPSPNQPTKHGDNREHPNEQ