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Target
TSC22 domain family protein 3
Ligand
BDBM50354850
Substrate
n/a
Meas. Tech.
GILZ gene assays
IC50
0.900±n/a nM
Citation
 Garbaccio, RM; Kern, JC; Mulhearn, JJ; Brandish, PE Phosphonate linkers and their use to facilitate cellular retention of compounds US Patent  US10869929 Publication Date 12/22/2020 
Target
Name:
TSC22 domain family protein 3
Synonyms:
DSIP-immunoreactive peptide | DSIPI | Delta sleep-inducing peptide immunoreactor | GILZ | Glucocorticoid-induced leucine zipper protein | Protein DIP | T22D3_HUMAN | TSC-22-like protein | TSC-22-related protein | TSC-22R | TSC22D3 | hDIP
Type:
Protein
Mol. Mass.:
14799.51
Organism:
Human
Description:
Q99576
Residue:
134
Sequence:
MNTEMYQTPMEVAVYQLHNFSISFFSSLLGGDVVSVKLDNSASGASVVAIDNKIEQAMDLVKNHLMYAVREEVEILKEQIRELVEKNSQLERENTLLKTLASPEQLEKFQSCLSPEEPAPESPQVPEAPGGSAV
  
Inhibitor
Name:
BDBM50354850
Synonyms:
BUDESONIDE | US10869929, Compound Budesonide | US11554172, Compound Budesonide | US11760775, Compound Budesonide
Type:
Small organic molecule
Emp. Form.:
C25H34O6
Mol. Mass.:
430.5339
SMILES:
CCCC1O[C@@H]2C[C@H]3[C@@H]4CCC5=CC(=O)C=C[C@]5(C)[C@H]4[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO |r,c:15,t:11|
Structure:
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