Affinity DataKi: 0.600nMAssay Description:In vitro ability of the compound to inhibit the amidolytic activity of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:In vitro ability of the compound to inhibit the amidolytic activity of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:In vitro ability of the compound to inhibit the amidolytic activity of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:In vitro ability of the compound to inhibit the amidolytic activity of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:In vitro ability of the compound to inhibit the amidolytic activity of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:In vitro ability of the compound to inhibit the amidolytic activity of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 100nM ΔG°: -39.8kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:In vitro ability of the compound to inhibit the amidolytic activity of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 480nM ΔG°: -35.9kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 780nM ΔG°: -34.7kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:In vitro ability of the compound to inhibit the amidolytic activity of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:In vitro ability of the compound to inhibit the amidolytic activity of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:In vitro ability of the compound to inhibit the amidolytic activity of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nM ΔG°: -33.3kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nM ΔG°: -33.0kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nM ΔG°: -32.1kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nM ΔG°: -30.7kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nM ΔG°: -30.7kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 4.20E+3nM ΔG°: -30.6kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nM ΔG°: -30.5kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 4.70E+3nM ΔG°: -30.3kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 7.90E+3nM ΔG°: -29.0kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 7.90E+3nM ΔG°: -29.0kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nM ΔG°: -29.0kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nM ΔG°: -29.0kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 8.30E+3nM ΔG°: -28.9kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 8.30E+3nM ΔG°: -28.9kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 8.50E+3nM ΔG°: -28.8kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 8.50E+3nM ΔG°: -28.8kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 9.40E+3nM ΔG°: -28.6kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nM ΔG°: -28.4kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro ability of the compound to inhibit the amidolytic activity of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nM ΔG°: -27.8kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nM ΔG°: -27.6kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 4.20E+4nM ΔG°: -24.9kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 5.60E+4nM ΔG°: -24.2kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+4nM ΔG°: -24.0kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+5nM ΔG°: -22.3kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+5nM ΔG°: -21.8kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+5nM ΔG°: -21.4kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+5nM ΔG°: -21.0kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against ThrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of thrombin in rat plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of rat thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of rat thrombinMore data for this Ligand-Target Pair