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TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50652775BDBM50652775(CHEMBL4303308)
Affinity DataIC50: 1nMAssay Description:Inhibition of KDM4B (2 to 500 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50652776BDBM50652776(CHEMBL4786329)
Affinity DataIC50: 1nMAssay Description:Inhibition of KDM4B (2 to 500 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483927BDBM50483927(CHEMBL3183531)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of KDM4B (2 to 500 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513345BDBM50513345(CHEMBL4438830)
Affinity DataIC50: 4nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513343BDBM50513343(CHEMBL4449500)
Affinity DataIC50: 5nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513345BDBM50513345(CHEMBL4438830)
Affinity DataIC50: 6nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 195611BDBM195611(GSKJ1)
Affinity DataIC50: 7.30nMAssay Description:Inhibition of KDM4B (2 to 500 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513345BDBM50513345(CHEMBL4438830)
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513345BDBM50513345(CHEMBL4438830)
Affinity DataIC50: 8nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513343BDBM50513343(CHEMBL4449500)
Affinity DataIC50: 8nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50158844BDBM50158844(CHEMBL3785491)
Affinity DataIC50: 10nMAssay Description:Inhibition of human KDM4B (1 to 500 residues) measured by antibody-based fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50158844BDBM50158844(CHEMBL3785491)
Affinity DataIC50: 10nMAssay Description:Inhibition of human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using H3K4me3 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513343BDBM50513343(CHEMBL4449500)
Affinity DataIC50: 12nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513345BDBM50513345(CHEMBL4438830)
Affinity DataIC50: 12nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513372BDBM50513372(CHEMBL4440395)
Affinity DataIC50: 15nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50153092BDBM50153092(CHEMBL3775894)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513374BDBM50513374(CHEMBL4466130)
Affinity DataIC50: 18nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513352BDBM50513352(CHEMBL4592908)
Affinity DataIC50: 19nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513357BDBM50513357(CHEMBL4590283)
Affinity DataIC50: 20nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513348BDBM50513348(CHEMBL4585876)
Affinity DataIC50: 20nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513345BDBM50513345(CHEMBL4438830)
Affinity DataIC50: 21nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513343BDBM50513343(CHEMBL4449500)
Affinity DataIC50: 22nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513367BDBM50513367(CHEMBL4559561)
Affinity DataIC50: 24nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513361BDBM50513361(CHEMBL4567766)
Affinity DataIC50: 27nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50153093BDBM50153093(CHEMBL3775668)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513360BDBM50513360(CHEMBL4573390)
Affinity DataIC50: 29nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50151923BDBM50151923(CHEMBL3774537)
Affinity DataIC50: 31nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus-infected Sf9 cells using ARTKQTARK(Me3)STGGK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50151923BDBM50151923(CHEMBL3774537)
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513371BDBM50513371(CHEMBL4438034)
Affinity DataIC50: 32nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513344BDBM50513344(CHEMBL4447515)
Affinity DataIC50: 32nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513351BDBM50513351(CHEMBL4516101)
Affinity DataIC50: 33nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50598660BDBM50598660(CHEMBL5203308)
Affinity DataIC50: 33nMAssay Description:Inhibition of KDM4B (unknown origin) measured by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513349BDBM50513349(CHEMBL4561958)
Affinity DataIC50: 33nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 293660BDBM293660(3-({[(1S)-6-[methyl(phenyl)amino]-1,2,3,4-tetrahyd...)
Affinity DataIC50: 35nMAssay Description:Inhibition of KDM4B (unknown origin) using H3K9me3 as substrate and measured by LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50151919BDBM50151919(CHEMBL3775121)
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513343BDBM50513343(CHEMBL4449500)
Affinity DataIC50: 36nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513345BDBM50513345(CHEMBL4438830)
Affinity DataIC50: 36nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50151917BDBM50151917(CHEMBL3775548)
Affinity DataIC50: 39nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50153161BDBM50153161(CHEMBL3775545)
Affinity DataIC50: 39nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513346BDBM50513346(CHEMBL4525269)
Affinity DataIC50: 40nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50151921BDBM50151921(CHEMBL3774456)
Affinity DataIC50: 41nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513343BDBM50513343(CHEMBL4449500)
Affinity DataIC50: 43nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513366BDBM50513366(CHEMBL4435185)
Affinity DataIC50: 45nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513354BDBM50513354(CHEMBL4558689)
Affinity DataIC50: 47nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513362BDBM50513362(CHEMBL4520178)
Affinity DataIC50: 49nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50152029BDBM50152029(CHEMBL3775899)
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50153094BDBM50153094(CHEMBL3775277)
Affinity DataIC50: 55nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 293660BDBM293660(3-({[(1S)-6-[methyl(phenyl)amino]-1,2,3,4-tetrahyd...)
Affinity DataIC50: 56nMAssay Description:Inhibition of KDM4B (unknown origin) using biotinylated H3K9me3 peptide and alpha-ketoglutarate as substrate pretreated for 1 hr followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513375BDBM50513375(CHEMBL4464471)
Affinity DataIC50: 57nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
EpiTherapeutics Aps

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50153069BDBM50153069(CHEMBL3775953)
Affinity DataIC50: 61nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details Article
PubMed
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