Compile Data Set for Download or QSAR
Report error Found 1251 of affinity data for UniProtKB/TrEMBL: P00735
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM21745(2-[(1R,4S,7S,13S,19S,22S,25S,28S,31R,34S,40S,43S,4...)
Affinity DataKi: >2.50E+6nM ΔG°: >-14.7kJ/molepH: 8.5 T: 2°CAssay Description:The enzyme reaction was initiated by adding fluorescence peptide substrate to reaction mixture containing enzyme and test compounds. The enzyme activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2008
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50027292(3-(2,2,2-Trifluoro-acetyl)-1H-indole-6-carboxamidi...)
Affinity DataKi:  1.51E+6nMAssay Description:Inhibition constant against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50027296(3-Formyl-1H-indole-6-carboxamidine | CHEMBL317713)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition constant against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50027283(3-Acetyl-1H-indole-6-carboxamidine | CHEMBL321524)
Affinity DataKi:  1.89E+6nMAssay Description:Inhibition constant against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50067523(2-[2-(4-Carbamimidoyl-benzenesulfonylamino)-acetyl...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibitory activity against Thrombin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50067526(2-[2-(4-Carbamimidoyl-benzenesulfonylamino)-acetyl...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibitory activity against Thrombin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50041224((R)-3-(7-Carbamimidoyl-naphthalen-2-yl)-2-{4-[(S)-...)
Affinity DataKi: >2.00E+6nMAssay Description:Binding affinity towards Thrombin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50010023(CHEMBL145466)
Affinity DataKi: >1.00E+6nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50010024(CHEMBL3251530)
Affinity DataKi:  1.00E+6nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50010016(CHEMBL3251531)
Affinity DataKi:  1.00E+6nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50010017(CHEMBL353802)
Affinity DataKi: >1.00E+6nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50009926(CHEMBL3250026)
Affinity DataKi:  9.30E+5nMpH: 6.0Assay Description:Competitive inhibition of 16 X 10'-7 M bovine thrombin using Z-Lys-nitrophenyl ester as substrate incubated up to 1 hr at pH 6More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50038002(Benzamidine (Protonated) | CHEMBL537204 | CHEMBL20...)
Affinity DataKi:  8.90E+5nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM21742(2-[(1R,4S,7S,13S,19S,22S,25S,28S,31R,34S,40S,43S,4...)
Affinity DataKi:  8.27E+5nM ΔG°:  -17.4kJ/molepH: 8.5 T: 2°CAssay Description:The enzyme reaction was initiated by adding fluorescence peptide substrate to reaction mixture containing enzyme and test compounds. The enzyme activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2008
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50010026(CHEMBL3251193)
Affinity DataKi:  7.00E+5nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50010022(CHEMBL3251532)
Affinity DataKi:  3.00E+5nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50442066(CHEMBL2441034)
Affinity DataKi: >2.51E+5nMAssay Description:Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50442067(CHEMBL2441027)
Affinity DataKi: >2.51E+5nMAssay Description:Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50442067(CHEMBL2441027)
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50442066(CHEMBL2441034)
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50442097(CHEMBL2441059)
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50442098(CHEMBL2441061)
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50442101(CHEMBL2441063)
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50442102(CHEMBL2441065)
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50442063(CHEMBL2441026)
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50009977(CHEMBL484621)
Affinity DataKi:  2.00E+5nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50027289(3-Benzoyl-1H-indole-6-carboxamidine | CHEMBL102009)
Affinity DataKi:  1.76E+5nMAssay Description:Inhibition constant against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50532388(CHEMBL4441722)
Affinity DataKi:  1.73E+5nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50532388(CHEMBL4441722)
Affinity DataKi:  1.73E+5nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50027297(4-(5-Nitro-indol-1-ylmethyl)-benzamidine | CHEMBL1...)
Affinity DataKi:  1.64E+5nMAssay Description:Inhibition constant against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM21741(2-[(1R,4S,7S,13S,19S,22S,25S,28S,31R,34S,40S,43S,4...)
Affinity DataKi:  1.64E+5nM ΔG°:  -21.4kJ/molepH: 8.5 T: 2°CAssay Description:The enzyme reaction was initiated by adding fluorescence peptide substrate to reaction mixture containing enzyme and test compounds. The enzyme activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2008
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50292885(1-carbamimidoyl-N-(3-(4-fluorobenzyloxy)phenyl)pip...)
Affinity DataKi:  1.60E+5nMAssay Description:Inhibition of bovine factor 2a by amydolitic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50010020(CHEMBL167983)
Affinity DataKi:  1.58E+5nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50532392(CHEMBL4437656)
Affinity DataKi:  1.41E+5nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50532392(CHEMBL4437656)
Affinity DataKi:  1.41E+5nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50010014(CHEMBL3251529)
Affinity DataKi:  1.33E+5nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50029092(CHEMBL3343304)
Affinity DataKi:  1.33E+5nMAssay Description:Inhibition of bovine thrombin assessed as reduction in hydrolysis of chromogenic substrate S-2238 by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50010018(CHEMBL3251189)
Affinity DataKi:  1.08E+5nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50532397(CHEMBL4476627)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50532397(CHEMBL4476627)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50010027(CHEMBL145735)
Affinity DataKi: >1.00E+5nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50010019(CHEMBL145656)
Affinity DataKi:  7.90E+4nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50532400(CHEMBL4549153)
Affinity DataKi:  7.22E+4nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50532400(CHEMBL4549153)
Affinity DataKi:  7.22E+4nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50010015(CHEMBL388768 | 3,5-Bis(4-Amidinophenyl)Isoxazole)
Affinity DataKi:  6.62E+4nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50532395(CHEMBL4547050)
Affinity DataKi:  6.08E+4nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50532395(CHEMBL4547050)
Affinity DataKi:  6.08E+4nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50010010(CHEMBL3251533)
Affinity DataKi:  5.67E+4nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50027301(2-Propionyl-1H-indole-6-carboxamidine | CHEMBL3219...)
Affinity DataKi:  5.50E+4nMAssay Description:Inhibition constant against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Georgetown University Medical Center

LigandPNGBDBM50292894(N-(3-((2',4'-difluorobiphenyl-4-yl)methoxy)phenyl)...)
Affinity DataKi:  5.40E+4nMAssay Description:Inhibition of bovine factor 2a by amydolitic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
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