Compile Data Set for Download or QSAR
Report error Found 199 of affinity data for UniProtKB/TrEMBL: P06199
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50448377BDBM50448377(CHEMBL3121473)
Affinity DataEC50:  0.0794nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50448377BDBM50448377(CHEMBL3121473)
Affinity DataEC50:  0.166nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 86231BDBM86231(CAS_51-55-8 | NSC_3661 | Atropine,(-) | ATROPINE |...)
Affinity DataKi:  0.390nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 86231BDBM86231(CAS_51-55-8 | NSC_3661 | Atropine,(-) | ATROPINE |...)
Affinity DataKi:  0.680nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50225215BDBM50225215(N,N,N-triethyl-2-(3-(((6-(2-(1,2,3,4-tetrahydroacr...)
Affinity DataEC50:  0.900nMAssay Description:Inhibition of [3H]NMS dissociation from porcine muscarinic M2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371197BDBM50371197(CHEMBL555247)
Affinity DataEC50:  1nMAssay Description:Inhibition of [3H]NMS dissociation from porcine muscarinic M2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50225209BDBM50225209(N,N,N-triethyl-2-(4-(((6-(2-(1,2,3,4-tetrahydroacr...)
Affinity DataEC50:  1.30nMAssay Description:Inhibition of [3H]NMS dissociation from porcine muscarinic M2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50225210BDBM50225210(N,N,N-triethyl-2-(5-(((6-(2-(1,2,3,4-tetrahydroacr...)
Affinity DataEC50:  1.40nMAssay Description:Inhibition of [3H]NMS dissociation from porcine muscarinic M2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371199BDBM50371199(CHEMBL540132)
Affinity DataEC50:  1.5nMAssay Description:Inhibition of [3H]NMS dissociation from porcine muscarinic M2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 86231BDBM86231(CAS_51-55-8 | NSC_3661 | Atropine,(-) | ATROPINE |...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025038BDBM50025038(Alcuronium)
Affinity DataEC50:  2nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093896BDBM50093896(Caracurine V derivative | CHEMBL311649)
Affinity DataEC50:  3nMAssay Description:Allosteric inhibition of [3H]NMS (N-methyl-scopolamine) dissociation from porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093893BDBM50093893(Caracurine V derivative | CHEMBL433343)
Affinity DataEC50:  4nMAssay Description:Allosteric inhibition of [3H]NMS (N-methyl-scopolamine) dissociation from porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50448376BDBM50448376(Naphmethonium)
Affinity DataEC50:  4.40nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371198BDBM50371198(CHEMBL540131)
Affinity DataEC50:  5nMAssay Description:Inhibition of [3H]NMS dissociation from porcine muscarinic M2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50176065BDBM50176065(CHEMBL76897 | CHEMBL168067 | 4-Diphenylacetoxy-1,1...)
Affinity DataKi:  6.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50448375BDBM50448375(CHEMBL3121479)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474538BDBM50474538(CHEMBL406691)
Affinity DataEC50:  7.60nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474526BDBM50474526(CHEMBL269592)
Affinity DataEC50:  7.80nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50448374BDBM50448374(CHEMBL3121478)
Affinity DataEC50:  7.80nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025036BDBM50025036(CHEMBL3337858)
Affinity DataEC50:  8nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093891BDBM50093891(Caracurine V derivative | CHEMBL315340)
Affinity DataEC50:  8nMAssay Description:Allosteric inhibition of [3H]NMS (N-methyl-scopolamine) dissociation from porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474523BDBM50474523(CHEMBL8532)
Affinity DataEC50:  8.5nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50176065BDBM50176065(CHEMBL76897 | CHEMBL168067 | 4-Diphenylacetoxy-1,1...)
Affinity DataKi:  10.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025035BDBM50025035(CHEMBL3337859)
Affinity DataEC50:  11nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50448375BDBM50448375(CHEMBL3121479)
Affinity DataEC50:  11nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025031BDBM50025031(CHEMBL3337863)
Affinity DataEC50:  12nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50448372BDBM50448372(CHEMBL3121475)
Affinity DataEC50:  12nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025031BDBM50025031(CHEMBL3337863)
Affinity DataEC50:  12nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474535BDBM50474535(CHEMBL8721)
Affinity DataEC50:  14nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 80806BDBM80806(3-[1,3-bis(oxidanylidene)benzo[de]isoquinolin-2-yl...)
Affinity DataEC50:  14nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50448369BDBM50448369(CHEMBL3121476)
Affinity DataEC50:  14nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474536BDBM50474536(CHEMBL274564)
Affinity DataEC50:  19nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50448370BDBM50448370(CHEMBL3120178)
Affinity DataEC50:  19nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50448374BDBM50448374(CHEMBL3121478)
Affinity DataEC50:  21nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50448371BDBM50448371(CHEMBL3121480)
Affinity DataEC50:  21nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018056BDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  21.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474529BDBM50474529(CHEMBL8449)
Affinity DataEC50:  25nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018056BDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  28.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093899BDBM50093899(Caracurine V derivative | CHEMBL314491)
Affinity DataEC50:  30nMAssay Description:Allosteric inhibition of [3H]NMS (N-methyl-scopolamine) dissociation from porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025030BDBM50025030(CHEMBL3355097)
Affinity DataEC50:  32nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025030BDBM50025030(CHEMBL3355097)
Affinity DataEC50:  32nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473900BDBM50473900(CHEMBL124330)
Affinity DataEC50:  36nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025027BDBM50025027(CHEMBL3337867)
Affinity DataEC50:  36nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474524BDBM50474524(CHEMBL406431)
Affinity DataEC50:  36nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025027BDBM50025027(CHEMBL3337867)
Affinity DataEC50:  36nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50448373BDBM50448373(CHEMBL3121477)
Affinity DataEC50:  38nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474548BDBM50474548(CHEMBL609382)
Affinity DataEC50:  45nMAssay Description:Ability to dissociate radioligand [3H]NMS from muscarinic acetylcholine receptor M2 of porcine heartMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473899BDBM50473899(CHEMBL262632)
Affinity DataEC50:  47nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50448371BDBM50448371(CHEMBL3121480)
Affinity DataEC50:  47nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
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