Compile Data Set for Download or QSAR
Report error Found 52 of affinity data for UniProtKB/TrEMBL: P11308
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417421BDBM50417421(CHEMBL1290597)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417418BDBM50417418(CHEMBL1289617)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417417BDBM50417417(CHEMBL1289509)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417426BDBM50417426(CHEMBL1289721)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003336BDBM50003336(CHEMBL3234565)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003076BDBM50003076(CHEMBL3234574)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417419BDBM50417419(CHEMBL1289618)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417414BDBM50417414(CHEMBL1289276)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413549BDBM50413549(CHEMBL513715)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003334BDBM50003334(CHEMBL3234564)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417420BDBM50417420(CHEMBL1290486)
Affinity DataKi:  3.16E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003407BDBM50003407(CHEMBL3234568)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003477BDBM50003477(CHEMBL3234569)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417422BDBM50417422(CHEMBL1289048)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417409BDBM50417409(CHEMBL1290487)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417410BDBM50417410(CHEMBL1290596)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413550BDBM50413550(CHEMBL469345)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417416BDBM50417416(CHEMBL1287827)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417423BDBM50417423(CHEMBL1289164)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003286BDBM50003286(CHEMBL3234576)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003289BDBM50003289(CHEMBL3234578)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417425BDBM50417425(CHEMBL1289510)
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417415BDBM50417415(CHEMBL1289277)
Affinity DataKi:  7.94E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003287BDBM50003287(CHEMBL3234577)
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417427BDBM50417427(CHEMBL1290716)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417424BDBM50417424(CHEMBL1289394)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379275BDBM50379275(CHEMBL2011500)
Affinity DataKd:  1.17E+4nMAssay Description:Binding affinity to ERG by surface plasmon resonanceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50352421BDBM50352421(CHEMBL1823591)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 251922BDBM251922(US9475814, 22 | US10065961, Compound 22 | US106832...)
Affinity DataIC50: 1.20E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent

TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003283BDBM50003283(CHEMBL3234575)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50420920BDBM50420920(CHEMBL2087549 | CHEMBL2087567)
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibition of human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50081399BDBM50081399(US9475814, 19 | CHEMBL3422016 | US10065961, Compou...)
Affinity DataIC50: 1.70E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent

TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003563BDBM50003563(CHEMBL3234573)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003562BDBM50003562(CHEMBL3234572)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 251928BDBM251928(US9475814, 31 | US10065961, Compound 31 | US106832...)
Affinity DataIC50: 2.00E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent

TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003561BDBM50003561(CHEMBL3234571)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 251927BDBM251927(US9475814, 29 | US10065961, Compound 29 | US106832...)
Affinity DataIC50: 2.50E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent

TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417412BDBM50417412(CHEMBL1289047)
Affinity DataKi:  2.51E+4nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50081363BDBM50081363(US9475814, 3 | CHEMBL3422012 | US10065961, Compoun...)
Affinity DataIC50: 2.60E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent

TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50352420BDBM50352420(CHEMBL1823865)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50352296BDBM50352296(CHEMBL1822468)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003559BDBM50003559(CHEMBL3234570)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003573BDBM50003573(CHEMBL3234871)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003291BDBM50003291(CHEMBL3234579)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 251913BDBM251913(US9475814, 11 | US10065961, Compound 11 | US106832...)
Affinity DataIC50: 3.00E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent

TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 251906BDBM251906(US9475814, 4 | US10065961, Compound 4 | US10683295...)
Affinity DataIC50: 3.00E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent

TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 251905BDBM251905(US9475814, 2 | US10065961, Compound 2 | US10683295...)
Affinity DataIC50: 3.00E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent

TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50081195BDBM50081195(US9475814, 1 | CHEMBL3422010 | US10065961, Compoun...)
Affinity DataIC50: 3.00E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent

TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417413BDBM50417413(CHEMBL1289163)
Affinity DataKi:  3.16E+4nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetTranscriptional regulator ERG(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50417411BDBM50417411(CHEMBL1290715)
Affinity DataKi: >3.16E+4nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
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