Compile Data Set for Download or QSAR
Report error Found 31 of affinity data for UniProtKB/TrEMBL: P28088
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043326BDBM50043326(c(Cys-Ser-Cys)-Ser-Ser-Leu-Met-Asp-Lys-Gln-c(Cys-V...)
Affinity DataIC50: 0.0930nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000558BDBM50000558(Endothelin-1 | ET-1 | Endothelin -1 | c(Cys-Ser-c(...)
Affinity DataIC50: 0.120nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043322BDBM50043322(c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-V...)
Affinity DataIC50: 0.170nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368776BDBM50368776(CHEMBL1790962)
Affinity DataIC50: 0.170nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289647BDBM50289647(Compound RES-701-1(1-10)/[A15]ET-1 | CHEMBL263855)
Affinity DataIC50: 0.240nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368772BDBM50368772(CHEMBL2373291)
Affinity DataIC50: 0.25nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368774BDBM50368774(CHEMBL1790963)
Affinity DataIC50: 0.330nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368777BDBM50368777(CHEMBL2373292)
Affinity DataIC50: 0.420nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043324BDBM50043324(c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-V...)
Affinity DataIC50: 0.450nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289650BDBM50289650(Compound RES-701-1(1-10)/[A15]ET-3 | CHEMBL414047)
Affinity DataIC50: 2.5nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289648BDBM50289648(Compound RES-701-1(1-10)/[A15]SRTX6b | CHEMBL40843...)
Affinity DataIC50: 3.80nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289112BDBM50289112(RES-701-1-C-terminal analogue | CHEMBL438745)
Affinity DataIC50: 6.30nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289108BDBM50289108(RES-701-1 | RES-701-1-C-terminal analogue | CHEMBL...)
Affinity DataIC50: 7.30nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289108BDBM50289108(RES-701-1 | RES-701-1-C-terminal analogue | CHEMBL...)
Affinity DataIC50: 10nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289111BDBM50289111(RES-701-1-C-terminal analogue | CHEMBL411057)
Affinity DataIC50: 10nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289107BDBM50289107(RES-701-1-C-terminal analogue | CHEMBL263294)
Affinity DataIC50: 12nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289113BDBM50289113(RES-701-1-C-terminal analogue | CHEMBL267754)
Affinity DataIC50: 36nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289117BDBM50289117(RES-701-1-C-terminal analogue | CHEMBL407422)
Affinity DataIC50: 45nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289109BDBM50289109(RES-701-1-C-terminal analogue | CHEMBL409339)
Affinity DataIC50: 54nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289116BDBM50289116(RES-701-1-C-terminal analogue | CHEMBL441573)
Affinity DataIC50: 98nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289115BDBM50289115(RES-701-1-C-terminal analogue | CHEMBL410321)
Affinity DataIC50: 120nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289114BDBM50289114(RES-701-1-C-terminal analogue | CHEMBL409433)
Affinity DataIC50: 450nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289110BDBM50289110(RES-701-1-C-terminal analogue | CHEMBL414131)
Affinity DataIC50: 470nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289656BDBM50289656(RES-701-1 | CHEMBL416287)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289651BDBM50289651(Compound [S15]ET-1 | CHEMBL407188)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289653BDBM50289653(ET-1 | Endothelin 1 | Et 1 | ENDOTHELIN)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289657BDBM50289657(RES-701-1 | CHEMBL414168)
Affinity DataIC50: 3.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289652BDBM50289652(Compound ET-3 | CHEMBL437610)
Affinity DataIC50: 3.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289654BDBM50289654(Compound SRTX6b | CHEMBL436894)
Affinity DataIC50: 3.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289649BDBM50289649(linear peptide of RES-701-1 | CHEMBL429908)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50289655BDBM50289655(N-C cyclized RES-70I-1 | CHEMBL414740)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article