Affinity DataEC50: 3nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 3nMAssay Description:Binding affinity to Retinoic acid receptor RXR-gamma was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Dissociation constant for binding to Retinoid X receptor gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-gamma was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of [3H]9-cis-RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-gamma was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of [3H]9-cis-RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of [3H]9-cis-RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of [3H]9-cis-RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-gamma was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-gamma was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibition of [3H]9-cis-RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Binding affinity to Retinoic acid receptor RXR-gamma was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Effective concentration against retinoid receptor isoform (RXR gamma) expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 29nMAssay Description:Inhibition of [3H]9-cis-RA binding to baculovirus expressed retinoid receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 29nMAssay Description:Binding affinity to Retinoic acid receptor RXR-gamma was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataKd: 35nMAssay Description:Inhibition of [3H]9-cis-RA binding to baculovirus expressed retinoid receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 36nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 36nMAssay Description:Effective concentration against retinoid receptor isoform (RXR gamma) expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 39nMAssay Description:Binding affinity to Retinoic acid receptor RXR-gamma was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 42nMAssay Description:Transcriptional activation of CV-1 cells expressing murine Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 42nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Effective concentration against retinoid receptor isoform (RXR gamma) expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 44nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 44nMAssay Description:Inhibition of [3H]9-cis-RA binding to baculovirus expressed retinoid receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 47nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-gamma was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataEC50: 49nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 59nMAssay Description:Inhibition of [3H]9-cis-RA binding to baculovirus expressed retinoid receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 73nMAssay Description:Dissociation constant for binding to Retinoid X receptor gammaMore data for this Ligand-Target Pair
Affinity DataIC50: 85nMAssay Description:Inhibition of binding to murine Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 94nMAssay Description:Inhibition of [3H]9-cis-RA binding to baculovirus expressed retinoid receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 113nMAssay Description:Inhibition of [3H]9-cis-RA binding to baculovirus expressed retinoid receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 124nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 128nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair


3D Structure (crystal)




























