Compile Data Set for Download or QSAR
Report error Found 119 of affinity data for UniProtKB/TrEMBL: P30082
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104037(His-Ser-Gln-Gly-Lys-Phe-Thr-Ser-Glu-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 0.200nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104040(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 0.240nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50122102(3-Cyano-4-hydroxy-benzoic acid [1-(2,3,5,6-tetrame...)
Affinity DataIC50: 0.430nMAssay Description:In vitro binding affinity towards rat glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50110054(3-Cyano-4-hydroxy-benzoic acid [1-[4-(4-isopropyl-...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity against rat glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 1.5nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50051588(His-Ser-Gln-thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Tyr-Le...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 1.5nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 1.5nMAssay Description:inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 1.5nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 1.5nMAssay Description:Compound was tested for its ability to displace [125I]glucagon from the glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104030(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ly...)
Affinity DataIC50: 1.70nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50051586([des-His1,Tyr5,Glu9,D-Tyr10]glucagon-NH2 | CHEMBL4...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104039(His-Ser-Gln-Cys-Thr-Phe-Thr-Ser-Cys-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 3.60nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098563(Ser-Gln-Gly-Thr-Phe-Thr-Ser-Glu-Tyr-Ser-Lys-Tyr-Le...)
Affinity DataIC50: 3.75nMAssay Description:Compound was evaluated for its ability to displace radiolabeled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50407844(CHEMBL2115191)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataEC50:  5nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in rat hepatocytes after 15 mins by cAMP dynamic2 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104031(His-Cys-Gln-Gly-Thr-Phe-Cys-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 5.60nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104043(His-Ser-Lys-Gly-Thr-Phe-Glu-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 6nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059362([des-His1, des-Phe6, Glu9] glucagon-NH2 | CHEMBL26...)
Affinity DataKd:  6.31nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104041(His-Ser-Gln-Gly-Thr-Phe-Cys-Ser-Asp-Tyr-Ser-Cys-Ty...)
Affinity DataIC50: 6.40nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataEC50:  8nMAssay Description:cAMP accumulation in rat hepatocytes in the presence rolipramMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50454201(CHEMBL3037804)
Affinity DataIC50: 10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104033(His-Ser-Gln-Gly-Thr-Phe-Lys-Ser-Asp-Tyr-Glu-Lys-Ty...)
Affinity DataIC50: 14nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104044(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 14nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098573(N-trinitrophenyl-His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-A...)
Affinity DataIC50: 15nMAssay Description:Compound was evaluated for its ability to displace radiolabeled glucagon (inactive up to 100 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059352([des-His1, Trp6, Glu9] glucagon-NH2 | CHEMBL442499)
Affinity DataIC50: 19nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098566(phenylbutyryl-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg-Arg-...)
Affinity DataIC50: 21.2nMAssay Description:IC50 value was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50171817(3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50: 23nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104096(3-Chloro-4-hydroxy-benzoic acid (4-hydroxy-naphtha...)
Affinity DataIC50: 27nMAssay Description:Binding affinity towards rat Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50557261(CHEMBL4749279)
Affinity DataEC50:  30nMAssay Description:Agonist activity at rat glucagon receptor expressed in HEK293 cells assessed as stimulation of cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098572(Ac-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg...)
Affinity DataIC50: 31nMAssay Description:IC50 value was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50407842(CHEMBL2114176)
Affinity DataIC50: 34.5nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50202031(3-(4-((1-(4-cyclohexenylphenyl)-3-(3,5-dichlorophe...)
Affinity DataIC50: 36nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059358([des-His1, Tyr6,Glu9] glucagon-NH2 | CHEMBL267885)
Affinity DataIC50: 40nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50244455((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3,5-dichl...)
Affinity DataIC50: 43nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059356([des-His1, Nle6, Glu9] glucagon-NH2 | CHEMBL236999...)
Affinity DataIC50: 48nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059362([des-His1, des-Phe6, Glu9] glucagon-NH2 | CHEMBL26...)
Affinity DataIC50: 48nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50284992(H-Ser-Gln-GlyThr-Thr-Ser-Glu-Tyr-Ser-Lys-Leu-Asp--...)
Affinity DataIC50: 48nMAssay Description:Compound was tested for its ability to displace [125I]glucagon from the glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098570(Ser-Gln-Gly-Thr-Thr-Ser-Glu-Tyr-Ser-Lys-Tyr-Leu-As...)
Affinity DataIC50: 48nMAssay Description:Compound was evaluated for its ability to displace radiolabeled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059359([des-His1, des-Gly4, Glu9] glucagon-NH2 | CHEMBL41...)
Affinity DataIC50: 52nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50087848(c[Asp15, Lys18,] glucagon-NH2 | CHEMBL427644)
Affinity DataIC50: 54nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50144009(3-{4-[1-(4-tert-Butyl-cyclohexyl)-3-(4-trifluorome...)
Affinity DataIC50: 56nMAssay Description:Inhibition of rat glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098565(Ac-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg-Arg-Ala-Gln-Asp...)
Affinity DataIC50: 60nMAssay Description:IC50 value was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50051585([des-His1,Tyr5,Glu9,(2S,3R)-beta-MePhe10]glucagon-...)
Affinity DataIC50: 74nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104036(His-Ser-Gln-Cys-Thr-Phe-Thr-Ser-Cys-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 85nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50057824(CHEMBL3326175)
Affinity DataIC50: 87nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059364([des-His1, D-Phe6, Glu9] glucagon-NH2 | CHEMBL2369...)
Affinity DataIC50: 100nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104032(His-Cys-Gln-Gly-Thr-Phe-Cys-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 101nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50611795(CHEMBL5277926)
Affinity DataIC50: 110nMAssay Description:Displacement of [125I]-glucagon from GCGR in Sprague-Dawley rat liver assessed as decrease in glucagon-stimulated CAMP production incubated for 45 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
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