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Report error Found 144 of affinity data for UniProtKB/TrEMBL: P35396
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50332462(2-(2-methyl-4-((4-methyl-2-(4-(trifluoromethyl)phe...)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at mouse PPAR-delta expressed in african green monkey CV-1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312479(2-(4-((4-(6-Morpholinopyridin-3-yl)-5-(4-(trifluor...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615952(CHEMBL5267473)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615955(CHEMBL5283926)
Affinity DataEC50:  6.10nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615962(CHEMBL5272996)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615966(CHEMBL5289740)
Affinity DataEC50:  6.90nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615954(CHEMBL5290870)
Affinity DataEC50:  6.90nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312476({4-[4-(6-Isopropoxypyridin-3-yl)-5-(4-trifluoromet...)
Affinity DataEC50:  7nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615964(CHEMBL5277165)
Affinity DataEC50:  7.5nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50539514(CHEMBL4649683)
Affinity DataEC50:  7.90nMAssay Description:Modulator activity at mouse PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312422(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312421(2-(4-((4-(4-Isopropoxyphenyl)-5-(4-(trifluorometho...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50383371(CHEMBL2030550)
Affinity DataIC50: 9.5nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312478(2-(4-((4-(2-Isopropoxypyrimidin-5-yl)-5-(4-(triflu...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615963(CHEMBL5290260)
Affinity DataEC50:  12nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615947(CHEMBL5278892)
Affinity DataEC50:  12nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312475(2-(4-((4-(6-Isopropoxypyridin-3-yl)-5-(4-(trifluor...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50619047(CHEMBL5424744)
Affinity DataEC50:  14nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50619057(CHEMBL5413218)
Affinity DataEC50:  14nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50619049(CHEMBL5416699)
Affinity DataEC50:  16nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312469(2-(4-((4-(4-Isopropoxyphenyl)-5-(4-propylphenyl)th...)
Affinity DataEC50:  17nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50619062(CHEMBL5432412)
Affinity DataEC50:  18nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50106105(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(4-tr...)
Affinity DataEC50:  19nMAssay Description:Agonist activity against PPAR deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50619045(CHEMBL5438357)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataEC50:  20nMAssay Description:Activity against murine PPAR delta receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50584465(CHEMBL5084377)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse PPARdelta in Cos7 cells transfected with pBIND and pGL4.35 Gal4 UAS Luc reporter plasmid by measuring luciferase activity i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312467(2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-isopropo...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50619055(CHEMBL5434437)
Affinity DataEC50:  22nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50085040({3-Chloro-4-[3-(3-phenyl-7-propyl-benzofuran-6-ylo...)
Affinity DataEC50:  23nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615960(CHEMBL5289017)
Affinity DataEC50:  24nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615946(CHEMBL5271479)
Affinity DataEC50:  25nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615961(CHEMBL5268424)
Affinity DataEC50:  26nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50619048(CHEMBL5422049)
Affinity DataEC50:  26nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312424({4-[4-(4-Isopropoxyphenyl)-5-(4-trifluoromethoxyph...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50383371(CHEMBL2030550)
Affinity DataIC50: 26.9nMAssay Description:Displacement of fluormone Pan-PPAR Green from mouse recombinant GST-tagged PPARbeta/delta LBD after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615951(CHEMBL5285352)
Affinity DataEC50:  27nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50619061(CHEMBL5406333)
Affinity DataEC50:  28nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615958(CHEMBL5279586)
Affinity DataEC50:  28nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312470(2-(4-((4-(4-Isopropoxyphenyl)-5-(4-biphenyl)thiazo...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50619050(CHEMBL5423281)
Affinity DataEC50:  29nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312472(2-(4-((5-(4-Biphenyl)-4-(pyridin-3-yl)oxazol-2-yl)...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312477(2-(4-((4-(2-Methoxypyrimidin-5-yl)-5-(4-propylphen...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50127222({4-[2-(3-Fluoro-4-trifluoromethyl-phenyl)-4-methyl...)
Affinity DataEC50:  30nMAssay Description:Activity against murine PPAR delta receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312425(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Affinity DataEC50:  31nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50619044(CHEMBL5431819)
Affinity DataEC50:  33nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50619054(CHEMBL5426189)
Affinity DataEC50:  33nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615957(CHEMBL5268646)
Affinity DataEC50:  34nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50619060(CHEMBL5412146)
Affinity DataEC50:  34nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615959(CHEMBL5273427)
Affinity DataEC50:  39nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50619052(CHEMBL5431069)
Affinity DataEC50:  41nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
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