Compile Data Set for Download or QSAR
Report error Found 15 of affinity data for UniProtKB/TrEMBL: P48302
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304497BDBM50304497(2-(5-{[4-(Benzo[1,3]dioxol-5-yl)-2-hydroxy-2-(4-me...)
Affinity DataKi:  1.26nMAssay Description:Displacement of [125I]ET1 from endothelin B receptor in DBA mouse microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50336697BDBM50336697(3-Benzo[1,3]dioxol-5-yl-4-[3-(2-{2-[2-(2-{4-[4-(2-...)
Affinity DataKi:  37nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304499BDBM50304499(3-Benzo[1,3]dioxol-5-yl-5-hydroxy-5-[4-(2-bromoeth...)
Affinity DataKi:  72nMAssay Description:Displacement of [125I]ET1 from endothelin B receptor in DBA mouse microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304495BDBM50304495(2-{4-[4-(Benzo[1,3]dioxol-5-yl)-2-hydroxy-5-oxo-3-...)
Affinity DataKi:  96nMAssay Description:Displacement of [125I]ET1 from endothelin B receptor in DBA mouse microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304498BDBM50304498(3-Benzo[1,3]dioxol-5-yl-5-[4-(2-fluoroethoxy)pheny...)
Affinity DataKi:  98nMAssay Description:Displacement of [125I]ET1 from endothelin B receptor in DBA mouse microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304494BDBM50304494(3-Benzo[1,3]dioxol-5-yl-4-[3-(2-bromoethoxy)-4,5-d...)
Affinity DataKi:  170nMAssay Description:Displacement of [125I]ET1 from endothelin B receptor in DBA mouse microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304496BDBM50304496(3-Benzo[1,3]dioxol-5-yl-4-[3-(2-fluoroethoxy)-4,5-...)
Affinity DataKi:  240nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304496BDBM50304496(3-Benzo[1,3]dioxol-5-yl-4-[3-(2-fluoroethoxy)-4,5-...)
Affinity DataKi:  240nMAssay Description:Displacement of [125I]ET1 from endothelin B receptor in DBA mouse microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50336699BDBM50336699(N-[1-(2-{2-[2-(2-{5-[4-Benzo[1,3]dioxol-5-yl-2-hyd...)
Affinity DataKi:  288nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50336694BDBM50336694(3-Benzo[1,3]dioxol-5-yl-4-{3-(2-(2-(2-(2-fluoroeth...)
Affinity DataKi:  418nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50034267BDBM50034267(PD156707 | PD-156707 | CHEMBL8981 | 3-Benzo[1,3]di...)
Affinity DataIC50: 780nMAssay Description:Displacement of [125I]ET1 from endothelin B receptor in DBA mouse microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50336698BDBM50336698(N-[1-(2-{2-[2-(2-{5-[4-Benzo[1,3]dioxol-5-yl-2-hyd...)
Affinity DataKi:  893nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50336696BDBM50336696(3-Benzo[1,3]dioxol-5-yl-4-[3-(2-{2-[2-(2-{1-[2-(2-...)
Affinity DataKi:  5.34E+3nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50336700BDBM50336700(3-Benzo[1,3]dioxol-5-yl-4-{3-[2-(2-{2-[2-(4-fluoro...)
Affinity DataKi:  6.45E+3nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetEndothelin receptor type B(Mouse)
University Hospital M£Nster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50336695BDBM50336695(3-Benzo[1,3]dioxol-5-yl-4-{3-[1-(2-{2-[2-(2-fluoro...)
Affinity DataKi:  8.45E+3nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed