Compile Data Set for Download or QSAR
Report error Found 16 of affinity data for UniProtKB/TrEMBL: Q14995
TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 643177BDBM643177(US20240002380, Example 3)
Affinity DataIC50: 250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 643178BDBM643178(US20240002380, Example 4)
Affinity DataIC50: 250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 643191BDBM643191(US20240002380, Example 45)
Affinity DataIC50: 250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 643199BDBM643199(US20240002380, Example 59)
Affinity DataIC50: 250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 643190BDBM643190(US20240002380, Example 44)
Affinity DataIC50: 250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 643181BDBM643181(US20240002380, Example 10)
Affinity DataIC50: 250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 50366239BDBM50366239(CHEMBL1961797)
Affinity DataIC50: 560nMAssay Description:Increased REV-ERB-beta LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 50366238BDBM50366238(CHEMBL1961796)
Affinity DataIC50: 800nMAssay Description:Increased REV-ERB-beta LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 643179BDBM643179(US20240002380, Example 5)
Affinity DataIC50: 1.00E+3nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 50095837BDBM50095837(CHEMBL3590573)
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of REV-ERBbeta (unknown origin) expressed in HEK293 cells incubated for 24 hrs assessed as inhibition of receptor-mediated transcriptional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 643192BDBM643192(US20240002380, Example 46)
Affinity DataIC50: 1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 643188BDBM643188(US20240002380, Example 34)
Affinity DataIC50: 1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 643201BDBM643201(US20240002380, Example 68)
Affinity DataIC50: 1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 643197BDBM643197(US20240002380, Example 56)
Affinity DataIC50: 1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 643195BDBM643195(US20240002380, Example 51)
Affinity DataIC50: 1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 2(Human)
Saint Louis University

US Patent
LigandChemical structure of BindingDB Monomer ID 50095836BDBM50095836(CHEMBL3590544)
Affinity DataIC50: 1.75E+4nMAssay Description:Inhibition of REV-ERBbeta (unknown origin) expressed in HEK293 cells incubated for 24 hrs assessed as inhibition of receptor-mediated transcriptional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed