Compile Data Set for Download or QSAR
Report error Found 146 of affinity data for UniProtKB/TrEMBL: Q6QHF9
LigandChemical structure of BindingDB Monomer ID 50015358BDBM50015358(N,N'-BIS(2,3-BUTADIENYL)-1,4-BUTANE-DIAMINE | CHEM...)
Affinity DataKi:  90nMAssay Description:Inhibitory activity measured as apparent dissociation constant against Polyamine oxidase (PAO) from pig liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50405943BDBM50405943(CHEMBL176596)
Affinity DataKi:  96nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50405931BDBM50405931(CHEMBL367753)
Affinity DataKi:  100nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 152706BDBM152706(Chlorhexidine (1) | Chlorhexidine)
Affinity DataKi:  100nM ΔG°:  -40.0kJ/molepH: 7.5 T: 2°CAssay Description:The APAO and SMO activities were measured spectrophotometrically by following the formation of a pink adduct (ε515 nm = 2.6 × 10^4 M−1 cm&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50405937BDBM50405937(CHEMBL173782)
Affinity DataKi:  180nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50026232BDBM50026232(N-Buta-2,3-dienyl-N'-methyl-butane-1,4-diamine | C...)
Affinity DataKi:  300nMAssay Description:Inhibitory activity measured as apparent dissociation constant against Polyamine oxidase (PAO) from pig liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50405942BDBM50405942(CHEMBL175345)
Affinity DataKi:  630nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50026231BDBM50026231(N*1*-Buta-2,3-dienyl-butane-1,4-diamine | CHEMBL59...)
Affinity DataKi:  700nMAssay Description:Inhibitory activity measured as apparent dissociation constant against Polyamine oxidase (PAO) from pig liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50405939BDBM50405939(CHEMBL175307)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50018055BDBM50018055(CHEMBL176843 | 7-Amino-heptan-2-one)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 741191BDBM741191(US20250161307, Example 34)
Affinity DataIC50: 1.10E+4nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741183BDBM741183(US20250161307, Example 26)
Affinity DataIC50: 2.20E+4nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50405932BDBM50405932(CHEMBL176530)
Affinity DataKi:  2.60E+4nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50405935BDBM50405935(CHEMBL177305)
Affinity DataKi:  3.10E+4nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 741182BDBM741182(US20250161307, Example 25)
Affinity DataIC50: 3.50E+4nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741184BDBM741184(US20250161307, Example 27)
Affinity DataIC50: 4.90E+4nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50405928BDBM50405928(CHEMBL174669)
Affinity DataKi:  7.50E+4nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 741185BDBM741185(US20250161307, Example 28)
Affinity DataIC50: 8.50E+4nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741274BDBM741274(US20250161307, Example 118)
Affinity DataIC50: 1.03E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50405940BDBM50405940(CHEMBL177890)
Affinity DataKi:  1.10E+5nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 741272BDBM741272(US20250161307, Example 116)
Affinity DataIC50: 1.19E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741238BDBM741238(US20250161307, Example 81)
Affinity DataIC50: 1.23E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741187BDBM741187(US20250161307, Example 30)
Affinity DataIC50: 1.29E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50405930BDBM50405930(CHEMBL174887)
Affinity DataKi:  1.30E+5nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 741257BDBM741257(US20250161307, Example 101)
Affinity DataIC50: 1.81E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741273BDBM741273(US20250161307, Example 117)
Affinity DataIC50: 1.97E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741271BDBM741271(US20250161307, Example 115)
Affinity DataIC50: 2.13E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741169BDBM741169(US20250161307, Example 12)
Affinity DataIC50: 2.33E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50405934BDBM50405934(CHEMBL176764)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 741237BDBM741237(US20250161307, Example 80)
Affinity DataIC50: 2.89E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741239BDBM741239(US20250161307, Example 82)
Affinity DataIC50: 2.91E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741177BDBM741177(US20250161307, Example 20)
Affinity DataIC50: 3.06E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741176BDBM741176(US20250161307, Example 19)
Affinity DataIC50: 3.07E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50026230BDBM50026230(N-Methyl-N'-prop-2-ynyl-butane-1,4-diamine | CHEMB...)
Affinity DataKi:  3.10E+5nMAssay Description:Inhibitory activity measured as apparent dissociation constant against Polyamine oxidase (PAO) from pig liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 741192BDBM741192(US20250161307, Example 35)
Affinity DataIC50: 3.62E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50405929BDBM50405929(CHEMBL436093)
Affinity DataKi:  3.76E+5nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 741244BDBM741244(US20250161307, Example 87)
Affinity DataIC50: 3.87E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741104BDBM741104(US20250161307, Example 1)
Affinity DataIC50: 3.97E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50026233BDBM50026233(N*1*-Prop-2-ynyl-butane-1,4-diamine | CHEMBL292770)
Affinity DataKi:  4.25E+5nMAssay Description:Inhibitory activity measured as apparent dissociation constant against Polyamine oxidase (PAO) from pig liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 741265BDBM741265(US20250161307, Example 109)
Affinity DataIC50: 4.70E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741262BDBM741262(US20250161307, Example 106)
Affinity DataIC50: 4.85E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741249BDBM741249(US20250161307, Example 92)
Affinity DataIC50: 5.20E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741179BDBM741179(US20250161307, Example 22)
Affinity DataIC50: 5.35E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741234BDBM741234(US20250161307, Example 77)
Affinity DataIC50: 5.44E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741259BDBM741259(US20250161307, Example 103)
Affinity DataIC50: 5.47E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741277BDBM741277(US20250161307, Example 121)
Affinity DataIC50: 6.41E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741250BDBM741250(US20250161307, Example 93)
Affinity DataIC50: 6.43E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50405941BDBM50405941(CHEMBL177777)
Affinity DataKi:  6.50E+5nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 741261BDBM741261(US20250161307, Example 105)
Affinity DataIC50: 6.66E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 741175BDBM741175(US20250161307, Example 18)
Affinity DataIC50: 6.80E+5nMAssay Description:The hPAOX assay was run and the data analyzed similarly to the hSMOX assay described above, except the reactions contained 60 pM recombinant PAOX wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

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