Compile Data Set for Download or QSAR
Report error Found 181 for UniProtKB: Q8VBU5
LigandChemical structure of BindingDB Monomer ID 14361BDBM14361(Adeo | 4-(3-cyclopentyloxy-4-methoxy-phenyl)pyrrol...)
Affinity DataIC50: 4nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2018
Entry Details
PDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 14361BDBM14361(Adeo | 4-(3-cyclopentyloxy-4-methoxy-phenyl)pyrrol...)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2018
Entry Details
PDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50213340BDBM50213340(CHEMBL58915)
Affinity DataIC50: 32nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50213338BDBM50213338(CHEMBL294883)
Affinity DataIC50: 78nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50213341BDBM50213341(CHEMBL59269)
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50213339BDBM50213339(CHEMBL291537)
Affinity DataIC50: 220nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2018
Entry Details

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140174BDBM140174(US8901315, 382)
Affinity DataIC50: 620nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140086BDBM140086(US8901315, 165)
Affinity DataIC50: 650nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140173BDBM140173(US8901315, 381)
Affinity DataIC50: 670nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140099BDBM140099(US8901315, 188)
Affinity DataIC50: 700nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140079BDBM140079(US8901315, 150)
Affinity DataIC50: 700nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140095BDBM140095(US8901315, 179)
Affinity DataIC50: 750nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140128BDBM140128(US8901315, 256)
Affinity DataIC50: 810nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140097BDBM140097(US8901315, 181)
Affinity DataIC50: 860nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140085BDBM140085(US8901315, 163)
Affinity DataIC50: 900nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140177BDBM140177(US8901315, 396)
Affinity DataIC50: 900nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140169BDBM140169(US8901315, 375)
Affinity DataIC50: 930nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140101BDBM140101(US8901315, 191)
Affinity DataIC50: 980nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140088BDBM140088(US8901315, 167)
Affinity DataIC50: 1.00E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140051BDBM140051(US8901315, 73)
Affinity DataIC50: 1.00E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140065BDBM140065(US8901315, 109)
Affinity DataIC50: 1.00E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140098BDBM140098(US8901315, 184)
Affinity DataIC50: 1.10E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140171BDBM140171(US8901315, 379)
Affinity DataIC50: 1.20E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140050BDBM140050(US8901315, 72)
Affinity DataIC50: 1.20E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140068BDBM140068(US8901315, 112)
Affinity DataIC50: 1.20E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140063BDBM140063(US8901315, 107 | US8901315, 106)
Affinity DataIC50: 1.20E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140142BDBM140142(US8901315, 275)
Affinity DataIC50: 1.20E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140087BDBM140087(US8901315, 166)
Affinity DataIC50: 1.30E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140090BDBM140090(US8901315, 170)
Affinity DataIC50: 1.30E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140184BDBM140184(US8901315, 416)
Affinity DataIC50: 1.30E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140060BDBM140060(US8901315, 101)
Affinity DataIC50: 1.30E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140096BDBM140096(US8901315, 180)
Affinity DataIC50: 1.40E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140108BDBM140108(US8901315, 203)
Affinity DataIC50: 1.40E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140126BDBM140126(US8901315, 247)
Affinity DataIC50: 1.40E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140176BDBM140176(US8901315, 395)
Affinity DataIC50: 1.40E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140089BDBM140089(US8901315, 168)
Affinity DataIC50: 1.50E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140172BDBM140172(US8901315, 380)
Affinity DataIC50: 1.50E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140069BDBM140069(US8901315, 367 | US8901315, 368 | US8901315, 114)
Affinity DataIC50: 1.50E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140070BDBM140070(US8901315, 115)
Affinity DataIC50: 1.50E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140081BDBM140081(US8901315, 155)
Affinity DataIC50: 1.50E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140062BDBM140062(US8901315, 104)
Affinity DataIC50: 1.50E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140140BDBM140140(US8901315, 273)
Affinity DataIC50: 1.60E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140083BDBM140083(US8901315, 366 | US8901315, 365 | US8901315, 159)
Affinity DataIC50: 1.60E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140075BDBM140075(US8901315, 141)
Affinity DataIC50: 1.60E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140094BDBM140094(US8901315, 177)
Affinity DataIC50: 1.60E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140100BDBM140100(US8901315, 190)
Affinity DataIC50: 1.70E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140091BDBM140091(US8901315, 171)
Affinity DataIC50: 1.70E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140141BDBM140141(US8901315, 274)
Affinity DataIC50: 1.70E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140093BDBM140093(US8901315, 176)
Affinity DataIC50: 1.70E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

TargetPhosphodiesterase(Mouse)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 140022BDBM140022(US8901315, 10)
Affinity DataIC50: 1.80E+3nMpH: 6.5 T: 2°CAssay Description:The PDE 4 (phosphodiesterase IV) inhibiting effect of the compounds of the present invention was performed by the following method, which was modifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
US Patent

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