Affinity DataKi: 0.0900nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M3 was determined in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M3 was determined in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 0.126nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.398nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Affinity DataIC50: 0.410nMAssay Description:Antagonist activity at M3 receptor in Dunkin-Hartley guinea pig tracheal strips assessed as inhibition of electrically field-stimulated contractile r...More data for this Ligand-Target Pair
Affinity DataIC50: 0.501nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M3 was determined in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 0.794nMAssay Description:Antagonism in muscarinic M3 receptor in guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataEC50: <1nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: <1nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: <1nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 1.30nMAssay Description:Antagonism in muscarinic M3 receptor in guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.53nMAssay Description:Antagonist activity at M3 receptor in Dunkin-Hartley guinea pig tracheal strips assessed as inhibition of electrically field-stimulated contractile r...More data for this Ligand-Target Pair
Affinity DataKd: 1.60nMAssay Description:Antagonism in muscarinic M3 receptor in guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Affinity DataEC50: 2.40nMAssay Description:In vitro contraction of guinea pig myenteric plexus preparation (mediated by Muscarinic M3 receptor)More data for this Ligand-Target Pair
Affinity DataKd: 2.5nMAssay Description:Antagonism in muscarinic M3 receptor in guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataKd: 2.5nMAssay Description:Antagonism in muscarinic M3 receptor in guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataIC50: 3.48nMAssay Description:Antagonist activity at M3 receptor in Dunkin-Hartley guinea pig tracheal strips assessed as inhibition of electrically field-stimulated contractile r...More data for this Ligand-Target Pair
Affinity DataIC50: 3.87nMAssay Description:Antagonist activity at M3 receptor in Dunkin-Hartley guinea pig tracheal strips assessed as inhibition of electrically field-stimulated contractile r...More data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Antagonism in muscarinic M3 receptor in guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at muscarinic M3 receptor in guinea pig trachea assessed as bronchorelaxation activity in presence of propranololMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Antagonist activity at M3 receptor in Dunkin-Hartley guinea pig tracheal strips assessed as inhibition of electrically field-stimulated contractile r...More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:In vitro binding affinity against guinea pig ileum using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
Affinity DataEC50: 5.30nMAssay Description:Agonist activity at muscarinic M3 receptor in guinea pig trachea assessed as bronchorelaxation activity in presence of propranololMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:In vitro binding affinity against guinea pig ileum using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Antagonism in muscarinic M3 receptor in guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:In vitro contraction of guinea pig myenteric plexus preparation (mediated by muscarinic acetylcholine receptor M3)More data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:In vitro contraction of guinea pig myenteric plexus preparation (mediated by Muscarinic M3 receptor)More data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:In vitro contraction of guinea pig myenteric plexus preparation (mediated by Muscarinic M3 receptor)More data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Antagonism in muscarinic M3 receptor in guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataKd: 32nMAssay Description:Antagonism in muscarinic M3 receptor in guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:In vitro binding affinity against guinea pig ileum using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:In vitro binding affinity against guinea pig ileum using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:In vitro binding affinity against guinea pig ileum using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
Affinity DataKd: 50nMAssay Description:Antagonism in muscarinic M3 receptor in guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:In vitro binding affinity against guinea pig ileum using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M3 was determined in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 79nMAssay Description:Antagonism in muscarinic M3 receptor in guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M3 was determined by measuring its ability to displace [3H]-N-methyl- Scopolamine...More data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:In vitro binding affinity against guinea pig ileum using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
Affinity DataKd: 91nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair












































