Compile Data Set for Download or QSAR
Report error Found 7 of affinity data for UniProtKB/TrEMBL: Q9JJX6
TargetP2X purinoceptor 4(Mouse)
Bayer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50506158BDBM50506158(CHEMBL4521594)
Affinity DataIC50: 112nMAssay Description:Antagonist activity at mouse P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of Mg-ATP-induced calcium influx incubated for 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetP2X purinoceptor 4(Mouse)
Bayer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50446060BDBM50446060(CHEMBL3103385)
Affinity DataIC50: 1.49E+4nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Mouse)
Bayer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50446072BDBM50446072(CHEMBL3103369)
Affinity DataIC50: 9.84E+4nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Mouse)
Bayer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50446076BDBM50446076(CHEMBL1483754)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Mouse)
Bayer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50446068BDBM50446068(CHEMBL3103375)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Mouse)
Bayer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50446070BDBM50446070(CHEMBL3103371)
Affinity DataIC50: 1.02E+5nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Mouse)
Bayer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50446069BDBM50446069(CHEMBL3103372)
Affinity DataIC50: 1.23E+5nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed