Compile Data Set for Download or QSAR
Report error Found 11 of affinity data for UniProtKB/TrEMBL: Q9Z286
TargetAdenylate cyclase type 10(Rat)
Tri-Institutional Institutional Therapeutics Discovery Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607676BDBM50607676(CHEMBL5218698 | US20240239774, Example 78)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of rat ADCY10 overexpressed in rat 4-4 cells assessed as IBMX stimulated cAMP accumulation preincubated for 10 mins followed by IBMX stimu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetAdenylate cyclase type 10(Rat)
Tri-Institutional Institutional Therapeutics Discovery Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607682BDBM50607682(CHEMBL5220685 | US20240239774, Example 139)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of rat ADCY10 overexpressed in rat 4-4 cells assessed as IBMX stimulated cAMP accumulation preincubated for 10 mins followed by IBMX stimu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetAdenylate cyclase type 10(Rat)
Tri-Institutional Institutional Therapeutics Discovery Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607686BDBM50607686(CHEMBL5219830 | US20240239774, Example 133)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of rat ADCY10 overexpressed in rat 4-4 cells assessed as IBMX stimulated cAMP accumulation preincubated for 10 mins followed by IBMX stimu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetAdenylate cyclase type 10(Rat)
Tri-Institutional Institutional Therapeutics Discovery Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607678BDBM50607678(CHEMBL5218878 | US20240239774, Example 76)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of rat ADCY10 overexpressed in rat 4-4 cells assessed as IBMX stimulated cAMP accumulation preincubated for 10 mins followed by IBMX stimu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetAdenylate cyclase type 10(Rat)
Tri-Institutional Institutional Therapeutics Discovery Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607685BDBM50607685(CHEMBL5220647 | US20240239774, Example 141)
Affinity DataIC50: 11nMAssay Description:Inhibition of rat ADCY10 overexpressed in rat 4-4 cells assessed as IBMX stimulated cAMP accumulation preincubated for 10 mins followed by IBMX stimu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetAdenylate cyclase type 10(Rat)
Tri-Institutional Institutional Therapeutics Discovery Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607679BDBM50607679(CHEMBL5218615 | US20240239774, Example 80)
Affinity DataIC50: 15nMAssay Description:Inhibition of rat ADCY10 overexpressed in rat 4-4 cells assessed as IBMX stimulated cAMP accumulation preincubated for 10 mins followed by IBMX stimu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetAdenylate cyclase type 10(Rat)
Tri-Institutional Institutional Therapeutics Discovery Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607680BDBM50607680(CHEMBL5218702 | US20240239774, Example 77)
Affinity DataIC50: 17nMAssay Description:Inhibition of rat ADCY10 overexpressed in rat 4-4 cells assessed as IBMX stimulated cAMP accumulation preincubated for 10 mins followed by IBMX stimu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetAdenylate cyclase type 10(Rat)
Tri-Institutional Institutional Therapeutics Discovery Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607681BDBM50607681(CHEMBL5218552 | US20240239774, Example 140)
Affinity DataIC50: 20nMAssay Description:Inhibition of rat ADCY10 overexpressed in rat 4-4 cells assessed as IBMX stimulated cAMP accumulation preincubated for 10 mins followed by IBMX stimu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetAdenylate cyclase type 10(Rat)
Tri-Institutional Institutional Therapeutics Discovery Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607684BDBM50607684(CHEMBL5219443 | US20240239774, Example 137)
Affinity DataIC50: 23nMAssay Description:Inhibition of rat ADCY10 overexpressed in rat 4-4 cells assessed as IBMX stimulated cAMP accumulation preincubated for 10 mins followed by IBMX stimu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetAdenylate cyclase type 10(Rat)
Tri-Institutional Institutional Therapeutics Discovery Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607683BDBM50607683(CHEMBL5219579 | US20240239774, Example 132)
Affinity DataIC50: 35nMAssay Description:Inhibition of rat ADCY10 overexpressed in rat 4-4 cells assessed as IBMX stimulated cAMP accumulation preincubated for 10 mins followed by IBMX stimu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetAdenylate cyclase type 10(Rat)
Tri-Institutional Institutional Therapeutics Discovery Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607677BDBM50607677(CHEMBL5220632 | US20240239774, Example 95)
Affinity DataIC50: 38nMAssay Description:Inhibition of rat ADCY10 overexpressed in rat 4-4 cells assessed as IBMX stimulated cAMP accumulation preincubated for 10 mins followed by IBMX stimu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed