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BindingDB contains 3.2M data for 1.4M Compounds and 11.5K Targets. Of those, 1.6M data for 780K Compounds and 4.8K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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64 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
7
New dermatological agents for the treatment of psoriasis.EBI
Allergan
4
Synthesis and pharmacologic evaluation of 2-endo-amino-3-exo-isopropylbicyclo[2.2.1]heptane: a potent imidazoline1 receptor specific agent.EBI
Allergan
7
Synthesis and biological activity of retinoic acid receptor-alpha specific amides.EBI
Allergan
4
Enantioselective syntheses of potent retinoid X receptor ligands: differential biological activities of individual antipodes.EBI
Allergan
9
Phenylcyclohexene and phenylcyclohexadiene substituted compounds having retinoid antagonist activity.EBI
Allergan
6
A new class of potent RAR antagonists: dihydroanthracenyl, benzochromenyl and benzothiochromenyl retinoids.EBI
Allergan
4
Stereoselective synthesis and receptor activity of conformationally defined retinoid X receptor selective ligands.EBI
Allergan
16
High affinity retinoic acid receptor antagonists: analogs of AGN 193109.EBI
Allergan
14
Synthesis and evaluation of 2-(arylamino)imidazoles as alpha 2-adrenergic agonists.EBI
Allergan
4
Identification of retinoic acid receptor beta subtype specific agonists.EBI
Allergan
8
Synthesis and structure-activity relationships of retinoid X receptor selective diaryl sulfide analogs of retinoic acid.EBI
Allergan
5
Synthesis and evaluation of 2-[(5-methylbenz-1-ox-4-azin-6-yl)imino]imidazoline, a potent, peripherally acting alpha 2 adrenoceptor agonist.EBI
Allergan
5
Identification of a retinoic acid receptor alpha subtype specific agonist.EBI
Allergan
15
Synthesis and carbonic anhydrase inhibitory activity of 4-substituted 2-thiophenesulfonamides.EBI
Allergan
10
Synthesis and structure-activity relationships of stilbene retinoid analogs substituted with heteroaromatic carboxylic acids.EBI
Allergan
2
Synthesis and characterization of a highly potent and effective antagonist of retinoic acid receptors.EBI
Allergan
6
Identification of highly potent retinoic acid receptor alpha-selective antagonists.EBI
Allergan
2
Conformational control in structure-based drug design.EBI
Allergan
119
3,4-disubstituted 3-cyclobutene-1,2-diones and use thereofBDB
Allergan
41
Imidazole derivatives as formyl peptide receptor modulatorsBDB
Allergan
179
Use of agonists of formyl peptide receptor 2 for treating dermatological diseasesBDB
Allergan
72
Pyridyl benzothiophenes as kinase inhibitorsBDB
Allergan
72
Pyridyl benzothiophenes as kinase inhibitorsBDB
Allergan
179
Use of agonists of formyl peptide receptor 2 for treating dermatological diseasesBDB
Allergan
13
Heterocycle-substituted pyridyl benzothiophenes as kinase inhibitorsBDB
Allergan
41
Imidazole derivatives as formyl peptide receptor modulatorsBDB
Allergan
72
Pyridyl benzothiophenes as kinase inhibitorsBDB
Allergan
88
Method of treating conditions with kinase inhibitorsBDB
Allergan
187
Use of agonists of formyl peptide receptor 2 for treating ocular inflammatory diseasesBDB
Allergan
146
Compounds as tyrosine kinase modulatorsBDB
Allergan
209
Sulfur derivatives as chemokine receptor modulatorsBDB
Allergan
11
Pharmaceutical compositions and methods of use of 4-pregenen-11β-17-21-triol-3,20-dione derivativesBDB
Allergan
26
1,2- bis-sulfonamide derivatives as chemokine receptor modulatorsBDB
Allergan
13
Heterocycle-substituted pyridyl benzothiophenes as kinase inhibitorsBDB
Allergan
5
Coumarin compounds as receptor modulators with therapeutic utilityBDB
Allergan
25
Substituted nicotinamide derivatives as kinase inhibitorsBDB
Allergan
38
Cyclosporins modified on the MeBmt sidechain by heterocyclic ringsBDB
Allergan
24
Compounds and methods for skin repairBDB
Allergan
19
15-aryl prostaglandins as EP4 agonists, and methods of use thereofBDB
Allergan
33
Cannabinoid-2 agonistsBDB
Allergan
83
Substituted 6,7-dialkoxy-3-isoquinolinol derivatives as inhibitors of phosphodiesterase 10 (PDE 10A)BDB
Allergan
10
Indole-3-carboxamides as kinase inhibitorsBDB
Allergan
16
Therapeutic prostaglandin receptor agonistsBDB
Allergan
7
Substituted 1,2,3,4-tetrahydropyrido[3,4-E] pyrrolo[1,2-A]pyrimidines as kinaseBDB
Allergan
87
Method of treating conditiions with kinase inhibitorsBDB
Allergan
25
Kinase inhibitorsBDB
Allergan
26
Indole-1-carboxamides as kinase inhibitorsBDB
Allergan
69
Compounds as tyrosine kinase modulatorsBDB
Allergan
1
Compounds and methods for treating ocular diseasesBDB
Allergan
5
Kinase inhibitorsBDB
Allergan
7
Kinase inhibitorsBDB
Allergan
17
Piperidylpyrimidine derivatives as modulators of protein kinase inhibitors and of vascular endothelial growth factor receptor 2BDB
Allergan
42
Substituted dialkyl(oxido)-lambda4-sulfanylidene nicotinamide derivatives as kinase inhibitorsBDB
Allergan
8
Substituted 1,2,3,4-tetrahydrobenzo[C][2,7] naphthyridines and derivatives thereof as kinase inhibitorsBDB
Allergan
30
Kinase inhibitorsBDB
Allergan
167
Substituted 6, 7-dialkoxy-3-isoquinoline derivatives as inhibitors of phosphodiesterase 10 (PDE 10A)BDB
Allergan
22
Treatment of inflammatory bowel diseaseBDB
Allergan
36
Cannabinoid-2 agonistsBDB
Allergan
29
3-phenyl-5-ureidoisothiazole-4-carboximide and 3-amino-5-phenylisothiazole derivatives as kinase inhibitorsBDB
Allergan
88
Kinase inhibitorsBDB
Allergan
84
Substituted 6,7-dialkoxy-3-isoquinolinol derivatives as inhibitors of phosphodiesterase 10 (PDE10A)BDB
Allergan
146
Compounds as tyrosine kinase modulatorsBDB
Allergan
16
S1P3 receptor inhibitors for treating painBDB
Allergan
154
6-substituted indole-3-carboxylic acid amide compounds having sphingosine-1-phosphate (S1P) receptor antagonist biological activityBDB
Allergan