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17 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis, in vitro evaluation and cocrystal structure of 4-oxo-[1]benzopyrano[4,3-c]pyrazole Cryptosporidium parvum inosine 5'-monophosphate dehydrogenase (CpIMPDH) inhibitors.EBI
University of Houston
Binding of curcumin and its long chain derivatives to the activator binding domain of novel protein kinase C.EBI
University of Houston
HIV-1 integrase pharmacophore model derived from diverse classes of inhibitors.EBI
University of Houston
Binding of isoxazole and pyrazole derivatives of curcumin with the activator binding domain of novel protein kinase C.EBI
University of Houston
Chemical modifications of resveratrol for improved protein kinase C alpha activity.EBI
University of Houston
Linker optimization and activity validation of a cell surface vimentin targeted homo-dimeric peptoid antagonist for lung cancer stem cells.EBI
University of Houston
Dynamic pharmacophore model optimization: identification of novel HIV-1 integrase inhibitors.EBI
University of Houston
Dynamic receptor-based pharmacophore model development and its application in designing novel HIV-1 integrase inhibitors.EBI
University of Houston
Design of pyrido[2,3-d]pyrimidin-7-one inhibitors of receptor interacting protein kinase-2 (RIPK2) and nucleotide-binding oligomerization domain (NOD) cell signaling.EBI
University of Houston
Receptor-interacting protein kinase 2 (RIPK2) and nucleotide-binding oligomerization domain (NOD) cell signaling inhibitors based on a 3,5-diphenyl-2-aminopyridine scaffold.EBI
University of Houston
Repurposing of Drugs-The Ketamine Story.EBI
University of Houston
Mycophenolic anilides as broad specificity inosine-5'-monophosphate dehydrogenase (IMPDH) inhibitors.EBI
University of Houston
Synthesis and activity of benzimidazole-1,3-dioxide inhibitors of separase.EBI
University of Houston
Discovery of covalent enzyme inhibitors using virtual docking of covalent fragments.EBI
University of Houston
Synthesis and activity of functionalizable derivatives of the serotonin (5-HT) 5-HTEBI
University of Houston
Activation loop targeting strategy for design of receptor-interacting protein kinase 2 (RIPK2) inhibitors.EBI
University of Houston
1-[2-(Diphenylmethoxy)ethyl]-2-methyl-5-nitroimidazole: a potent lead for the design of novel NNRTIs.BDB
Sapienza University of Rome