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9 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis and biological evaluation of a series of N-alkylated imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors.EBI
Ludwig-Maximilians-Universit£T M£Nchen
Straightforward and effective synthesis of¿-aminobutyric acid transporter subtype 2-selective acyl-substituted azaspiro[4.5]decanes.EBI
Universit£
Structure activity relationship of selective GABA uptake inhibitors.EBI
University of Copenhagen
First photoswitchable neurotransmitter transporter inhibitor: light-induced control of¿-aminobutyric acid transporter 1 (GAT1) activity in mouse brain.EBI
Ludwig-Maximilians-Universit£T M£Nchen
Synthesis, biological evaluation and structure-activity relationship of new GABA uptake inhibitors, derivatives of 4-aminobutanamides.EBI
Jagiellonian University Medical College
Selective mGAT2 (BGT-1) GABA uptake inhibitors: design, synthesis, and pharmacological characterization.EBI
University of Copenhagen
Nipecotic acid as potential lead molecule for the development of GABA uptake inhibitors; structural insights and design strategies.EBI
Isf College of Pharmacy
Development of tricyclic N-benzyl-4-hydroxybutanamide derivatives as inhibitors of GABA transporters mGAT1-4 with anticonvulsant, antinociceptive, and antidepressant activity.EBI
Jagiellonian University Medical College
Structure-Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/?-Aminobutyric Acid Transporter 1 (BGT1).EBI
University of Copenhagen