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15 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
(18)F-AmBF3-MJ9: a novel radiofluorinated bombesin derivative for prostate cancer imaging.EBI
Bc Cancer Agency
Studies toward the development of new silicon-containing building blocks for the direct (18)F-labeling of peptides.EBI
Institute of Technology (Eth) Zurich
Heterobivalent dual-target probe for targeting GRP and Y1 receptors on tumor cells.EBI
The Ohio State University
Targeting gastrin-releasing peptide receptors of prostate cancer cells for photodynamic therapy with a phthalocyanine-bombesin conjugate.EBI
Universit£
PD 176252--the first high affinity non-peptide gastrin-releasing peptide (BB2) receptor antagonist.EBI
Cambridge University Forvie Site
 
PD 165929 the first high affinity non-peptide neuromedin-B (NMB) receptor selective antagonistEBI
TBA
Discovery of MK-5046, a Potent, Selective Bombesin Receptor Subtype-3 Agonist for the Treatment of ObesityEBI
TBA
Synthesis and SAR of derivatives based on 2-biarylethylimidazole as bombesin receptor subtype-3 (BRS-3) agonists for the treatment of obesity.EBI
Merck Research Laboratories
Discovery of substituted biphenyl imidazoles as potent, bioavailable bombesin receptor subtype-3 agonists.EBI
Merck Research Laboratories
Discovery and optimization of a novel Neuromedin B receptor antagonist.EBI
Amgen
Structural assessment and biological evaluation of two N3S bombesin derivatives.EBI
Institutes of Radioisotopes-Radiodiagnostic Products and Biology
Discovery of small molecule agonists for the bombesin receptor subtype 3 (BRS-3) based on an omeprazole lead.EBI
Glaxosmithkline
Potent bombesin-like peptides for GRP-receptor targeting of tumors with 99mTc: a preclinical study.EBI
National Center For Scientific Research Demokritos
Design of selective peptidomimetic agonists for the human orphan receptor BRS-3.EBI
Technische UniversitäT MüNchen
Synthesis, Biological Evaluation, and Molecular Docking of 8-imino-2-oxo-2H,8H-pyrano[2,3-f]chromene Analogs: New Dual AChE Inhibitors as Potential Drugs for the Treatment of Alzheimer's Disease.BDB
Yogi Vemana University