PMID

Data

Article Title

Organization

Identification of novel class of falcipain-2 inhibitors as potential antimalarial agents.

University of Toronto

Synthesis of gallinamide A analogues as potent falcipain inhibitors and antimalarials.

The University of Sydney

Synthesis, antimalarial and antitubercular activity of acetylenic chalcones.

University of Cape Town

Constrained peptidomimetics as antiplasmodial falcipain-2 inhibitors.

Universit£

Development of peptidomimetics with a vinyl sulfone warhead as irreversible falcipain-2 inhibitors.

University of Messina

Identification of novel parasitic cysteine protease inhibitors using virtual screening. 1. The ChemBridge database.

University of Mississippi

Novel peptidomimetic cysteine protease inhibitors as potential antimalarial agents.

University of Messina

Identification of novel parasitic cysteine protease inhibitors by use of virtual screening. 2. The available chemical directory.

University of Mississippi

Design, synthesis and evaluation of 3-methylene-substituted indolinones as antimalarials.

University of Lisbon

Synthesis of novel peptidomimetics as inhibitors of protozoan cysteine proteases falcipain-2 and rhodesain.

University of Messina

Design and synthesis of novel 2-pyridone peptidomimetic falcipain 2/3 inhibitors.

University of Algarve

A prodomain peptide of Plasmodium falciparum cysteine protease (falcipain-2) inhibits malaria parasite development.

International Center For Genetic Engineering and Biotechnology

Design, synthesis, and antimalarial activity of structural chimeras of thiosemicarbazone and ferroquine analogues.

Université

Dipeptide vinyl sultams: synthesis via the Wittig-Horner reaction and activity against papain, falcipain-2 and Plasmodium falciparum.

University of Lisbon

Discovery of potent thiosemicarbazone inhibitors of rhodesain and cruzain.

University of California San Francisco

Synthesis and structure-activity relationships of parasiticidal thiosemicarbazone cysteine protease inhibitors against Plasmodium falciparum, Trypanosoma brucei, and Trypanosoma cruzi.

University of California San Francisco

Synthesis and evaluation of isatins and thiosemicarbazone derivatives against cruzain, falcipain-2 and rhodesain.

University of Cape Town

Identification of antimalarial leads with dual falcipain-2 and falcipain-3 inhibitory activity.

Shoolini University of Biotechnology and Management Sciences

Recent advances of tetrazole derivatives as potential anti-tubercular and anti-malarial agents.

Wuxi Apptec

Falcipain Inhibitors Based on the Natural Product Gallinamide A Are Potent in Vitro and in Vivo Antimalarials.

The University of Sydney

Synthesis and antimalarial effects of phenothiazine inhibitors of a Plasmodium falciparum cysteine protease.

Universidad Central De Venezuela

New aziridine-based inhibitors of cathepsin L-like cysteine proteases with selectivity for the Leishmania cysteine protease LmCPB2.8.

Johannes Gutenberg-Universit£T Mainz

Peptidomimetic nitrile inhibitors of malarial protease falcipain-2 with high selectivity against human cathepsins.

Irbm Science Park

Designing novel inhibitors against falcipain-2 of Plasmodium falciparum.

Delhi Institute of Pharmaceutical Sciences and Research

Quinoline hybrids and their antiplasmodial and antimalarial activities.

Hubei Engineering University

Development of Novel Peptide-Based Michael Acceptors Targeting Rhodesain and Falcipain-2 for the Treatment of Neglected Tropical Diseases (NTDs).

University of Messina

Synthesis and biological evaluation of phenolic Mannich bases of benzaldehyde and (thio)semicarbazone derivatives against the cysteine protease falcipain-2 and a chloroquine resistant strain of Plasmodium falciparum.

University of Cape Town

Synthesis and evaluation of new antimalarial phenylurenyl chalcone derivatives.

Universidad Central De Venezuela