BindingDB

The first public molecular recognition database, BindingDB supports research, education and practice in drug discovery, pharmacology and related fields.

BindingDB contains 3.2M data for 1.4M Compounds and 11.5K Targets. Of those, 1.6M data for 780K Compounds and 4.8K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

If BindingDB was of value to your research, please take a moment to donate to this nonprofit project. Your donation will let us provide you with more data and improved service.

Donate Now

To help with training and testing AI and other models, BindingDB downloads and search results now provide the publication date and BindingDB curation date of each measurement.

Advanced Search

24 articles for thisTarget

The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
4
Identification and characterization of a prostaglandin transporter.EBI
Albert Einstein College of Medicine
15
Estradiol 17 beta-D-glucuronide is a high-affinity substrate for oatp organic anion transporter.EBI
Albert Einstein College of Medicine
2
Cloning of mouse prostaglandin transporter PGT cDNA: species-specific substrate affinities.EBI
Albert Einstein College of Medicine
7
Identification of lactate as a driving force for prostanoid transport by prostaglandin transporter PGT.EBI
Albert Einstein College of Medicine
4
Structural determinants of substrates for the prostaglandin transporter PGT.EBI
Albert Einstein College of Medicine
2
Enzymatic transition states and dynamic motion in barrier crossing.EBI
Albert Einstein College of Medicine
1
Synthesis of novel ketoconazole derivatives as inhibitors of the human Pregnane X Receptor (PXR; NR1I2; also termed SXR, PAR).EBI
Albert Einstein College of Medicine
22
Transition State Analogs of Human DNPH1 Reveal Two Electrophile Migration Mechanisms.EBI
Albert Einstein College of Medicine
21
In Vivo-Active Soluble Epoxide Hydrolase-Targeting PROTACs with Improved Potency and Stability.EBI
Albert Einstein College of Medicine
10
Structural Insights into Protein-Inhibitor Interactions in Human Tryptophan Dioxygenase.EBI
Albert Einstein College of Medicine
13
Selective Inhibitors of Helicobacter pylori Methylthioadenosine Nucleosidase and Human Methylthioadenosine Phosphorylase.EBI
Albert Einstein College of Medicine
16
Current Insights of BRAF Inhibitors in Cancer.EBI
Albert Einstein College of Medicine
19
Compounds useful for inhibiting RAF dimersBDB
Albert Einstein College of Medicine
7
Heat Capacity Changes for Transition-State Analogue Binding and Catalysis with Human 5'-Methylthioadenosine Phosphorylase.BDB
Albert Einstein College of Medicine
10
Methods, assays and compounds for treating bacterial infections by inhibiting methylthioinosine phosphorylaseBDB
Albert Einstein College of Medicine
20
Transition state analogues of Plasmodium falciparum and human orotate phosphoribosyltransferases.BDB
Albert Einstein College of Medicine
2
High accuracy in silico sulfotransferase models.BDB
Albert Einstein College of Medicine
2
New IDH1 mutant inhibitors for treatment of acute myeloid leukemiaBDB
Albert Einstein College of Medicine
22
Altered enthalpy-entropy compensation in picomolar transition state analogues of human purine nucleoside phosphorylase.BDB
Albert Einstein College of Medicine
6
Kinetics and inhibition of nicotinamidase from Mycobacterium tuberculosis.BDB
Albert Einstein College of Medicine
2
Acyclic Immucillin Phosphonates: Second-Generation Inhibitors of Plasmodium falciparum Hypoxanthine- Guanine-Xanthine Phosphoribosyltransferase.BDB
Albert Einstein College of Medicine
10
Synthetic modification of prostaglandin f(2alpha) indicates different structural determinants for binding to the prostaglandin F receptor versus the prostaglandin transporter.BDB
Albert Einstein College of Medicine
8
Picomolar inhibitors as transition-state probes of 5'-methylthioadenosine nucleosidases.BDB
Albert Einstein College of Medicine
3
Transition state analogs of 5'-methylthioadenosine nucleosidase disrupt quorum sensing.BDB
Albert Einstein College of Medicine