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35 articles for thisTarget

The following articles (labelled with PubMed ID or TBD) are for your review

Article Title
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.EBI
Novel class of potent 4-arylalkyl substituted 3-isoxazolol GABA(A) antagonists: synthesis, pharmacology, and molecular modeling.EBI
The Royal Danish School of Pharmacy
Partial GABAA receptor agonists. Synthesis and in vitro pharmacology of a series of nonannulated analogs of 4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridin-3-ol.EBI
Royal Danish School of Pharmacy
3-Thienyl- and 3-furylaminobutyric acids. Synthesis and binding GABAB receptor studies.EBI
Laboratoire De Pharmacie Chimique, Facult�
Synthesis and biochemical evaluation of baclofen analogues locked in the baclofen solid-state conformation.EBI
Centre De Neurochimie Du Cnrs
GABA agonists and uptake inhibitors. Synthesis, absolute stereochemistry, and enantioselectivity of (R)-(-)- and (S)-(+)-homo-beta-proline.EBI
Royal Danish School of Pharmacy
Synthesis and pharmacological evaluation of gamma-aminobutyric acid analogues. New ligand for GABAB sites.EBI
Aminomethyl-2,6-difluorophenols as a novel class of increased lipophilicity GABA(C) receptor antagonists.EBI
The University of Sydney
The first selective antagonist for a GABAC receptorEBI
A study of 3-amino-N-hydroxypropanesulfonamide derivatives as potential GABAB agonists and their fragmentation to 3-aminopropanesulfinic acidEBI
Biological activity of 3-aminopropyl (methyl) phosphinic acid, a potent and selective GABAB agonist with CNS activityEBI
Synthesis and pharmacology of the baclofen homologues 5-amino-4-(4-chlorophenyl)pentanoic acid and the R- and S-enantiomers of 5-amino-3-(4-chlorophenyl)pentanoic acid.EBI
The Royal Danish School of Pharmacy
Phosphinic acid analogues of GABA. 2. Selective, orally active GABAB antagonists.EBI
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.EBI
Synthesis and activity of 5-(aminomethylene)-1,3-cyclohexanediones: enolic analogues of gamma-aminobutyric acid.EBI
Synthesis, Biological Evaluation, and Molecular Docking of 8-imino-2-oxo-2H,8H-pyrano[2,3-f]chromene Analogs: New Dual AChE Inhibitors as Potential Drugs for the Treatment of Alzheimer's Disease.BDB
Yogi Vemana University