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35 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.EBI
Universit£
Novel class of potent 4-arylalkyl substituted 3-isoxazolol GABA(A) antagonists: synthesis, pharmacology, and molecular modeling.EBI
The Royal Danish School of Pharmacy
Partial GABAA receptor agonists. Synthesis and in vitro pharmacology of a series of nonannulated analogs of 4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridin-3-ol.EBI
Royal Danish School of Pharmacy
3-Thienyl- and 3-furylaminobutyric acids. Synthesis and binding GABAB receptor studies.EBI
Laboratoire De Pharmacie Chimique, Facult�
Synthesis and biochemical evaluation of baclofen analogues locked in the baclofen solid-state conformation.EBI
Centre De Neurochimie Du Cnrs
GABA agonists and uptake inhibitors. Synthesis, absolute stereochemistry, and enantioselectivity of (R)-(-)- and (S)-(+)-homo-beta-proline.EBI
Royal Danish School of Pharmacy
Synthesis and pharmacological evaluation of gamma-aminobutyric acid analogues. New ligand for GABAB sites.EBI
TBA
Aminomethyl-2,6-difluorophenols as a novel class of increased lipophilicity GABA(C) receptor antagonists.EBI
The University of Sydney
 
The first selective antagonist for a GABAC receptorEBI
TBA
 
A study of 3-amino-N-hydroxypropanesulfonamide derivatives as potential GABAB agonists and their fragmentation to 3-aminopropanesulfinic acidEBI
TBA
 
Biological activity of 3-aminopropyl (methyl) phosphinic acid, a potent and selective GABAB agonist with CNS activityEBI
TBA
Synthesis and pharmacology of the baclofen homologues 5-amino-4-(4-chlorophenyl)pentanoic acid and the R- and S-enantiomers of 5-amino-3-(4-chlorophenyl)pentanoic acid.EBI
The Royal Danish School of Pharmacy
Phosphinic acid analogues of GABA. 2. Selective, orally active GABAB antagonists.EBI
Ciba-Geigy
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.EBI
Ciba-Geigy
Synthesis and activity of 5-(aminomethylene)-1,3-cyclohexanediones: enolic analogues of gamma-aminobutyric acid.EBI
TBA
Synthesis, Biological Evaluation, and Molecular Docking of 8-imino-2-oxo-2H,8H-pyrano[2,3-f]chromene Analogs: New Dual AChE Inhibitors as Potential Drugs for the Treatment of Alzheimer's Disease.BDB
Yogi Vemana University