BDBM50001157 CHEMBL538700
SMILES Cc1cc(O)cc(C)c1C[C@H](N)C(=O)N1Cc2ccccc2C[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(N)=O
InChI Key InChIKey=KYXSQGDWDGTJNF-BBACVFHCSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50001157
Affinity DataKi: 0.118nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal
Curated by ChEMBL
Clinical Research Institute of Montreal
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as induction of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair