BDBM25400 (2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol::CHEMBL68738::CPA::N6-CyclopentylAdo::N6-cyclopentyladenosine (CPA)::cid_657378
SMILES OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(NC3CCCC3)ncnc12
InChI Key InChIKey=SQMWSBKSHWARHU-SDBHATRESA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 25400
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.47E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.25E+3nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 16.9nMAssay Description:Agonist activity at adenosine A1 receptor in rat cortical membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in rat brain cortical membrane in absence of 100 uM GTPMore data for this Ligand-Target Pair
Affinity DataIC50: 154nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in rat brain cortical membrane in presence of 100 uM GTPMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR in absence of GTP by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 538nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR in presence of 100 uM of GTP by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR assessed as GTP shiftMore data for this Ligand-Target Pair