BDBM50324335 2'-Cyclohexylamino-6-((R)-pyrrolidin-3-ylamino)[2,4']bipyridinyl-4-carboxylic Acid Amide::CHEMBL1215220
SMILES NC(=O)c1cc(N[C@@H]2CCNC2)nc(c1)-c1ccnc(NC2CCCCC2)c1
InChI Key InChIKey=WXGCJNLWHYWDFU-QGZVFWFLSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50324335
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of PKD2 by TR-FRET assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase D1(Human)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+3nMAssay Description:Inhibition of PKD1 assessed as inhibition of HDAC5 neuclear exportMore data for this Ligand-Target Pair