BDBM264064 2-[5-[(6-chloro-1,2,3,4- tetrahydronaphthalen-1- yl)oxy]pyrazol-1-yl]pyridine-4- carboxylic acid::US10173996, Example 149::US9604961, Example 149::US9714230, 149::US9908865, Example 149
SMILES OC(=O)c1ccnc(c1)-n1nccc1OC1CCCc2cc(Cl)ccc12
InChI Key InChIKey=MYEIDQDVSWLKKZ-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 264064
Affinity DataIC50: 550nMAssay Description:The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...More data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction conditions: 0.8...More data for this Ligand-Target Pair