BDBM50079387 1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-piperidin-1-yl]-ethanol::CHEMBL28564::Eliprodil
SMILES OC(CN1CCC(Cc2ccc(F)cc2)CC1)c1ccc(Cl)cc1
InChI Key InChIKey=GGUSQTSTQSHJAH-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50079387
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory concentration against NMDA responses at NR1A/2C receptors expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory concentration against NMDA responses at cloned NR1A/2A receptors expressed in Xenopus oocytes More data for this Ligand-Target Pair
Affinity DataIC50: 277nMAssay Description:Displacement of [3H]-ifendropil from binding site of N-methyl-D-aspartate glutamate receptor was evaluated employing synaptosomal fraction of porcine...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Tested for the NMDA antagonist activity using a functional assay, by protection of cultured hippocampus neurons from the toxic effects of extracellul...More data for this Ligand-Target Pair
Affinity DataIC50: 1.13E+4nMAssay Description:Compound was tested for inhibition of [3H]-MK-801 binding to N-methyl-D-aspartate glutamate receptor lacking NR2B subunit in low affinity fraction of...More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Tested for the Alpha-1 adrenergic receptor affinity in a standard radioligand binding assay with [3H]- prazosinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibitory concentration against NMDA responses at NR1A/2B receptors expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Compound was tested for inhibition of [3H]-MK-801 binding to N-methyl-D-aspartate glutamate receptor at NR2B subunit in high affinity fraction of por...More data for this Ligand-Target Pair