BDBM50442757 CHEMBL2443026
SMILES CN(C)c1ccc(Oc2cc(O)cc(O)c2-c2cc(no2)C(=O)NC2CCN(CC2)C2CCC3(CC2)OCCO3)cc1
InChI Key InChIKey=DPZWKZQIGWCTDT-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 37 hits for monomerid = 50442757
Affinity DataIC50: >10nMAssay Description:Displacement of N6-(6-amino)hexyl-ATP ATTO-590-ATP from HSC70 (unknown origin) after 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of MST4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of MPS1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of MK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of MET (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of MELK (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of JAK3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of JAK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of IR (unknown origin)More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Nerviano Medical Sciences
Curated by ChEMBL
Nerviano Medical Sciences
Curated by ChEMBL
Affinity DataIC50: >10nMAssay Description:Inhibition of IKK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of IGFR1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of haspin (V473 to K798) (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of FAK (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of CK2alpha/beta (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of CHK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of ZAP70 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of TRKA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Nerviano Medical Sciences
Curated by ChEMBL
Nerviano Medical Sciences
Curated by ChEMBL
Affinity DataIC50: >10nMAssay Description:Inhibition of RET (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of PIM2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Nerviano Medical Sciences
Curated by ChEMBL
Nerviano Medical Sciences
Curated by ChEMBL
Affinity DataIC50: >10nMAssay Description:Inhibition of PERK (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of PDGFRbeta (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of PAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of CDC7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of BRK (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of Aurora kinase-2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of Aurora kinase-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of Alk (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of AKT1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of ACK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of NEK6 (unknown origin)More data for this Ligand-Target Pair