BDBM101478 US8524710, 55::US8530652, 49::US8530652, 5

SMILES CN(C)C[C@@H](NC(=O)N1Cc2c(Nc3ncnc4ccsc34)n[nH]c2C1(C)C)c1ccccc1

InChI Key InChIKey=CDSCKKVCQGIMOU-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 101478   

TargetSerine/threonine-protein kinase PAK 4(Human)
Agouron Pharmaceuticals

US Patent
LigandPNGBDBM101478(US8530652, 5 | US8530652, 49 | US8524710, 55)
Affinity DataKi:  220nM EC50:  87nMAssay Description:The enzymatic activity of PAK4 KD was measured by its ability to catalyzed the transfer of a phosphate residue from a nucleoside triphosphate to an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2013
Entry Details
US Patent