BDBM101728 US9695160, 30::US9796707, Compound 30

SMILES COc1ccc(CN2CCN(CC2)c2ccc(cc2NC(=O)c2ccc(o2)-c2ccncc2)C(F)(F)F)cc1

InChI Key InChIKey=WPGFUYWTZGYGSF-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 101728   

TargetSRSF protein kinase 1(Human)
The University of Nottingham

US Patent
LigandPNGBDBM101728(US9695160, 30 | US9796707, Compound 30)
Affinity DataIC50: 336nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetSRSF protein kinase 1(Human)
The University of Nottingham

US Patent
LigandPNGBDBM101728(US9695160, 30 | US9796707, Compound 30)
Affinity DataIC50: 336nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent