BDBM103932 US8569511, 16

SMILES CC(C)([N+]#[C-])c1ccc(cc1)-c1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1

InChI Key InChIKey=NWANDSBRGRLBGY-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 103932   

Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Utah

US Patent
LigandPNGBDBM103932(US8569511, 16)
Affinity DataIC50: 5.17E+3nMAssay Description:The secondary assay was a time resolved-FRET LanthaScreen Kinase Binding Assay. (Invitrogen Corporation, Carlsbad, Calif.). This assay evaluates the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2014
Entry Details
US Patent

Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Utah

US Patent
LigandPNGBDBM103932(US8569511, 16)
Affinity DataIC50: 5.85E+4nMAssay Description:The primary assay for compound inhibitory activity was the ATP depletion assay using the PDKtide substrate purchase from Millipore Corporation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2014
Entry Details
US Patent