BDBM103933 US8569511, 17

SMILES Fc1ccc(NC(=O)Nc2ccc3[nH]nc(-c4nc5ccccc5[nH]4)c3c2)c(F)c1

InChI Key InChIKey=HZUJMAYPJILNGE-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 103933   

Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Utah

US Patent
LigandPNGBDBM103933(US8569511, 17)
Affinity DataIC50: 1.00E+5nMAssay Description:The secondary assay was a time resolved-FRET LanthaScreen Kinase Binding Assay. (Invitrogen Corporation, Carlsbad, Calif.). This assay evaluates the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2014
Entry Details
US Patent

Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Utah

US Patent
LigandPNGBDBM103933(US8569511, 17)
Affinity DataIC50: 1.00E+5nMAssay Description:The primary assay for compound inhibitory activity was the ATP depletion assay using the PDKtide substrate purchase from Millipore Corporation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2014
Entry Details
US Patent