BDBM103936 US8569511, 20

SMILES O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCN(CC1)c1ccncc1

InChI Key InChIKey=NJXQUYNZYIQURR-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 103936   

Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Utah

US Patent
LigandPNGBDBM103936(US8569511, 20)
Affinity DataIC50: 1.00E+5nMAssay Description:The primary assay for compound inhibitory activity was the ATP depletion assay using the PDKtide substrate purchase from Millipore Corporation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2014
Entry Details
US Patent

Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Utah

US Patent
LigandPNGBDBM103936(US8569511, 20)
Affinity DataIC50: 1.00E+5nMAssay Description:The secondary assay was a time resolved-FRET LanthaScreen Kinase Binding Assay. (Invitrogen Corporation, Carlsbad, Calif.). This assay evaluates the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2014
Entry Details
US Patent