BDBM103937 US8569511, 21

SMILES FC1(F)CC1C(=O)Nc1ccc2c(n[nH]c2c1)-c1nc2ccc(cc2[nH]1)N1CCOCC1

InChI Key InChIKey=SEAWZPFSTWYPJA-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 103937   

Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Utah

US Patent
LigandPNGBDBM103937(US8569511, 21)
Affinity DataIC50: 1.00E+5nMAssay Description:The secondary assay was a time resolved-FRET LanthaScreen Kinase Binding Assay. (Invitrogen Corporation, Carlsbad, Calif.). This assay evaluates the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2014
Entry Details
US Patent

Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Utah

US Patent
LigandPNGBDBM103937(US8569511, 21)
Affinity DataIC50: 1.00E+5nMAssay Description:The primary assay for compound inhibitory activity was the ATP depletion assay using the PDKtide substrate purchase from Millipore Corporation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2014
Entry Details
US Patent