BDBM120528 US8703768, 128

SMILES CNC(=O)c1ncccc1NC(=O)c1nc(cnc1Nc1cncnc1)C1CC1

InChI Key InChIKey=GQGHTGUUCQIUIO-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 120528   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Hoffmann-La Roche

US Patent

LigandBDBM120528(US8703768, 128)Copy SMILESCopy InChI

Affinity DataIC50: 1.30nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
10/14/2014
Entry Details
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