BDBM137951 US8871934, 544

SMILES OC1(c2ccccc2-c2c1cc(F)cc2-c1cnn(CC2(O)CCCCC2)c1)C(F)(F)F

InChI Key InChIKey=DGXTXNBOWOYLBV-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 137951   

Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Human)
Japan Tobacco

US Patent

LigandBDBM137951(US8871934, 544)Copy SMILESCopy InChI

Affinity DataIC50: 22nMpH: 8.0 T: 2°CAssay Description:The inhibitory action of PDHK activity was indirectly evaluated by performing a kinase reaction in the presence of a test compound and measuring the ...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
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Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
4/6/2015
Entry Details
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